STAT6 Gain-of-Function Disease

Mendelian MONDO:0957807 Pathograph 18 Show in embeddings browser hereditary disease inborn error of immunity hyper-IgE syndrome

STAT6 gain-of-function (GOF) disease is a recently described autosomal dominant inborn error of immunity caused by germline heterozygous gain-of-function variants in STAT6, the transcription factor downstream of the type 2 cytokines IL-4 and IL-13. GOF variants (predominantly in the DNA-binding domain) cause constitutive/hyperresponsive STAT6 signaling with sustained phosphorylation, increased target-gene expression, and TH2 skewing, producing a profound early-life multisystem allergic phenotype: treatment-resistant atopic dermatitis, marked hypereosinophilia with eosinophilic gastrointestinal disease, asthma, very high serum IgE, IgE-mediated food allergy, and anaphylaxis, with variable susceptibility to infection. It is catalogued in OMIM as hyper-IgE syndrome 6 (HIES6). Type 2-directed therapy (the anti-IL-4Ra antibody dupilumab) and JAK inhibition (ruxolitinib) are effective targeted treatments.

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1
Inheritance
8
Pathophys.
15
Phenotypes
18
Pathograph
1
Genes
3
Medical Actions
1
References
1
Deep Research
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Classifications

Harrison's Part
IMMUNE RHEUMATOLOGIC GENETICS ENVIRONMENT DISEASE
IUIS Category
combined immunodeficiency with syndromic features
👪

Inheritance

1
Autosomal dominant inheritance HP:0000006
STAT6 GOF disease follows an autosomal dominant inheritance pattern from monoallelic (heterozygous) STAT6 variants; cases are either de novo/sporadic or transmitted through affected kindreds. Penetrance is complete, with variable expressivity.
Autosomal dominant inheritance Penetrance: COMPLETE Expressivity: VARIABLE
Show evidence (2 references)
PMID:36884218 SUPPORT Human Clinical
"The cases were either sporadic (seven kindreds) or followed an autosomal dominant inheritance pattern (three kindreds)."
Documents both sporadic/de novo and autosomal dominant transmission of heterozygous STAT6 GOF variants across the discovery cohort.
PMID:38238227 SUPPORT Human Clinical
"STAT6-GOF disease demonstrated complete penetrance, although some clinical variability"
The consortium review reports complete penetrance with clinical variability (variable expressivity).

Pathophysiology

8
STAT6 gain-of-function variant
Germline heterozygous rare variants in STAT6 (most in the DNA-binding domain, e.g. p.E372K, p.E377K) confer a gain of function: the mutant transcription factor shows increased DNA-binding affinity, a strong preference for nuclear localization, and spontaneous transcriptional activity.
STAT6 hgnc:11368 HUGO Gene Nomenclature Committee (hgnc) Relation: this pathophysiological event involves this gene This pathophysiological event involves STAT6 (hgnc:11368). hgnc:11368 is a gene from the HUGO Gene Nomenclature Committee.
Show evidence (2 references)
PMID:36884218 SUPPORT Human Clinical
"All patients carried monoallelic rare variants in STAT6 and functional studies established their gain-of-function (GOF) phenotype with sustained STAT6 phosphorylation, increased STAT6 target gene expression, and TH2 skewing."
Establishes monoallelic STAT6 variants with a functionally validated gain-of-function phenotype as the causal lesion.
PMID:36216080 SUPPORT Human Clinical
"We identified a heterozygous missense variant (c.1129G>A;p.Glu377Lys) in the DNA binding domain of STAT6 that was de novo in the index patient's father and was inherited by 2 of his 3 children."
Localizes a representative GOF variant to the STAT6 DNA-binding domain.
Constitutive STAT6 signaling
STAT6 is the central transcription factor of the type 2 cytokine (IL-4/IL-13) response. GOF variants produce sustained basal and cytokine-induced STAT6 phosphorylation and increased target-gene transcription, amplifying the allergic-inflammation program.
interleukin-4-mediated signaling pathway GO:0035771 Gene Ontology (GO) Relation: this pathophysiological event involves this biological process This pathophysiological event involves increased interleukin-4-mediated signaling pathway (GO:0035771). GO:0035771 is a biological process from the Gene Ontology. ↑ INCREASED JAK-STAT signaling GO:0007259 Gene Ontology (GO) Relation: this pathophysiological event involves this biological process This pathophysiological event involves increased JAK-STAT signaling, annotated with cell surface receptor signaling pathway via JAK-STAT (GO:0007259). GO:0007259 is a biological process from the Gene Ontology. ↑ INCREASED
Show evidence (5 references)
PMID:36884218 SUPPORT Human Clinical
"STAT6 (signal transducer and activator of transcription 6) is a transcription factor that plays a central role in the pathophysiology of allergic inflammation."
Establishes STAT6 as the central signaling node whose constitutive activity drives the disease.
PMID:36758835 SUPPORT In Vitro
"The mutation augmented both basal and cytokine-induced STAT6 phosphorylation without affecting dephosphorylation kinetics."
Functional assay of the mutated STAT6 protein documents increased basal and cytokine-induced STAT6 phosphorylation as the proximal signaling abnormality.
PMID:40603028 SUPPORT In Vitro
"even in the absence of IL-4 stimulation, we observed the translocation of mutant STAT6 in its unphosphorylated state, which activated gene expression."
Documents ligand- and phosphorylation-independent nuclear translocation of the D419N mutant, the most constitutive form of the signaling defect.
+ 2 more references
TH2 immune skewing
Constitutive STAT6 activity biases naive CD4+ T cells toward TH2 differentiation with elevated peripheral TH2 lymphocytes, producing the IL-4/ IL-5/IL-13-dominated milieu that underlies allergic effector disease.
T-helper 2 cell CL:0000546 Cell Ontology (CL) Relation: this pathophysiological event involves this cell type This pathophysiological event involves T-helper 2 cell (CL:0000546). CL:0000546 is a cell type from the Cell Ontology.
T-helper 2 cell differentiation GO:0045064 Gene Ontology (GO) Relation: this pathophysiological event involves this biological process This pathophysiological event involves increased T-helper 2 cell differentiation (GO:0045064). GO:0045064 is a biological process from the Gene Ontology. ↑ INCREASED
Show evidence (1 reference)
PMID:36216080 SUPPORT Human Clinical
"Higher levels of peripheral blood TH2 lymphocytes were detected."
Documents increased peripheral TH2 lymphocytes as the cellular readout of STAT6-driven skewing.
IgE class switching
The type 2 milieu drives B-cell immunoglobulin class switching to IgE, producing very high serum IgE — the humoral effector arm.
B cell CL:0000236 Cell Ontology (CL) Relation: this pathophysiological event involves this cell type This pathophysiological event involves B cell (CL:0000236). CL:0000236 is a cell type from the Cell Ontology.
isotype switching to IgE isotypes GO:0035708 Gene Ontology (GO) Relation: this pathophysiological event involves this biological process This pathophysiological event involves increased isotype switching to IgE isotypes, annotated with interleukin-4-dependent isotype switching to IgE isotypes (GO:0035708). GO:0035708 is a biological process from the Gene Ontology. ↑ INCREASED
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"hypereosinophilia with esosinophilic gastrointestinal disease, asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."
Documents elevated serum IgE (and IgE-mediated food allergy) as the humoral effector consequence of the type 2 program.
Eosinophil expansion
The type 2 milieu (IL-5) drives marked eosinophil expansion and tissue recruitment, producing blood hypereosinophilia and eosinophilic tissue infiltration — the cellular effector arm.
eosinophil CL:0000771 Cell Ontology (CL) Relation: this pathophysiological event involves this cell type This pathophysiological event involves eosinophil (CL:0000771). CL:0000771 is a cell type from the Cell Ontology.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"hypereosinophilia with esosinophilic gastrointestinal disease, asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."
Documents hypereosinophilia and eosinophilic gastrointestinal disease as the cellular effector consequence of the type 2 program.
Multisystem allergic disease
The convergent clinical endpoint: early-onset, treatment-resistant atopic dermatitis, asthma, eosinophilic gastrointestinal disease, IgE-mediated food allergy, and anaphylaxis.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"a profound phenotype of early-life onset allergic immune dysregulation, widespread treatment-resistant atopic dermatitis, hypereosinophilia with esosinophilic gastrointestinal disease, asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."
Enumerates the multisystem allergic phenotype that defines the disease.
Impaired antimicrobial immunity
Reciprocal suppression of TH1 and TH17 responses (the mirror image of TH2 skewing) impairs antimicrobial defense, underlying the recurrent skin, respiratory, and viral infections seen in a subset of patients and the OMIM designation of HIES6 as "with recurrent infections."
T-helper 1 cell CL:0000545 Cell Ontology (CL) Relation: this pathophysiological event involves this cell type This pathophysiological event involves T-helper 1 cell (CL:0000545). CL:0000545 is a cell type from the Cell Ontology. T-helper 17 cell CL:0000899 Cell Ontology (CL) Relation: this pathophysiological event involves this cell type This pathophysiological event involves T-helper 17 cell (CL:0000899). CL:0000899 is a cell type from the Cell Ontology.
T-helper 1 cell differentiation GO:0045063 Gene Ontology (GO) Relation: this pathophysiological event involves this biological process This pathophysiological event involves decreased T-helper 1 cell differentiation (GO:0045063). GO:0045063 is a biological process from the Gene Ontology. ↓ DECREASED T-helper 17 cell differentiation GO:0072539 Gene Ontology (GO) Relation: this pathophysiological event involves this biological process This pathophysiological event involves decreased T-helper 17 cell differentiation (GO:0072539). GO:0072539 is a biological process from the Gene Ontology. ↓ DECREASED
Show evidence (1 reference)
PMID:36758835 SUPPORT Human Clinical
"Naive lymphocytes from the affected patient displayed increased TH2- and suppressed TH1- and TH17-cell responses."
TH1/TH17 suppression provides the immunological basis for impaired antimicrobial defense.
B-cell lymphoma predisposition
STAT6 is a recurrently mutated oncogenic driver in follicular lymphoma and other B-cell lymphomas, and germline STAT6 GOF is associated with an emerging lymphoma risk: one reported patient developed follicular lymphoma that later relapsed as diffuse large B-cell lymphoma. The true magnitude of risk is not yet established.
B cell CL:0000236 Cell Ontology (CL) Relation: this pathophysiological event involves this cell type This pathophysiological event involves B cell (CL:0000236). CL:0000236 is a cell type from the Cell Ontology.
Show evidence (3 references)
PMID:38238227 SUPPORT Human Clinical
"To date, one patient found to have STAT6-GOF disease has developed lymphoma"
Documents the first reported lymphoma in a patient with germline STAT6 GOF disease.
PMID:38238227 SUPPORT Other
"STAT6 is frequently and recurrently mutated in follicular lymphomas and other B cell lymphomas"
Provides the biological rationale linking constitutive STAT6 activity to B-cell lymphomagenesis.
PMID:37316763 SUPPORT Human Clinical
"The clinical association of lymphoma in our kindred, along with previous data linking somatic STAT6 D419H mutations to follicular lymphoma suggest that patients with STAT6 GOF disease may be at higher risk of lymphomagenesis."
Independent kindred (germline p.D419H) directly linking STAT6 GOF disease to lymphoma risk, reinforcing the shared-residue rationale.

Pathograph

Use the checkboxes to hide or show graph categories. Hover nodes for evidence and cross-linked metadata.
Pathograph: causal mechanism network for STAT6 Gain-of-Function Disease Interactive directed graph showing how pathophysiology mechanisms, phenotypes, genetic factors and variants, experimental models, environmental triggers, and treatments relate through causal and linked edges.

Phenotypes

15
Blood 3
Increased circulating IgE concentration HP:0003212 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Increased circulating IgE concentration (HP:0003212). HP:0003212 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."
Documents elevated serum IgE as part of the core phenotype.
Eosinophilia Increased total eosinophil count HP:0001880 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Increased total eosinophil count (HP:0001880). HP:0001880 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:36758835 SUPPORT Human Clinical
"who presented with severe atopic dermatitis, eosinophilia, and elevated IgE."
Documents eosinophilia in an affected patient.
Lymphoma HP:0002665 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is B-cell lymphoma, annotated with Lymphoma (HP:0002665). HP:0002665 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"To date, one patient found to have STAT6-GOF disease has developed lymphoma"
Documents the first reported lymphoma in a patient with germline STAT6 GOF disease.
Cardiovascular 1
Lymphadenopathy HP:0002716 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Lymphadenopathy (HP:0002716). HP:0002716 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"Lymphoproliferation, characterized by lymphadenopathy"
Documents lymphadenopathy as a feature of STAT6 GOF lymphoproliferation.
Digestive 1
Gastroesophageal reflux HP:0002020 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Gastroesophageal reflux (HP:0002020). HP:0002020 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"gastroesophageal reflux disease"
Documents early gastroesophageal reflux disease as a diagnostic feature.
Immune 3
Atopic dermatitis HP:0001047 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Atopic dermatitis (HP:0001047), qualified as infantile onset. HP:0001047 is a phenotype from the Human Phenotype Ontology.
Onset: INFANTILE
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"a profound phenotype of early-life onset allergic immune dysregulation, widespread treatment-resistant atopic dermatitis"
Documents widespread treatment-resistant atopic dermatitis as a core feature.
Food allergy HP:0500093 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Food allergy (HP:0500093). HP:0500093 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:36216080 SUPPORT Human Clinical
"Severe atopic dermatitis and food allergy were key presentations."
Documents food allergy as a key presentation.
Recurrent infections HP:0002719 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Recurrent infections (HP:0002719). HP:0002719 is a phenotype from the Human Phenotype Ontology.
Show evidence (2 references)
PMID:38238227 SUPPORT Human Clinical
"with recurrent skin, respiratory, and viral infections, but no fatal infections were noted."
The consortium review documents recurrent skin, respiratory, and viral infections in a subset of patients.
PMID:36758835 SUPPORT Human Clinical
"Naive lymphocytes from the affected patient displayed increased TH2- and suppressed TH1- and TH17-cell responses."
TH1/TH17 suppression provides an immunological basis for infection susceptibility; recurrent infection is captured in the OMIM disease name.
Musculoskeletal 1
Osteoporosis HP:0000939 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Osteoporosis with pathological fractures, annotated with Osteoporosis (HP:0000939). HP:0000939 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"osteoporosis with pathological fractures, generalized joint"
Documents osteoporosis with pathological fractures as a reported feature.
Growth 1
Short stature HP:0004322 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Short stature (HP:0004322). HP:0004322 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"including short stature, pathological fractures,"
Documents short stature among the STAT3-LOF-overlapping non-immunological features of STAT6 GOF disease.
Other 5
Asthma HP:0002099 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Asthma (HP:0002099). HP:0002099 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"hypereosinophilia with esosinophilic gastrointestinal disease, asthma, elevated serum IgE"
Documents asthma as part of the phenotype.
Eosinophilic esophagitis Eosinophilic infiltration of the esophagus HP:0410151 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Eosinophilic esophagitis, annotated with Eosinophilic infiltration of the esophagus (HP:0410151). HP:0410151 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"hypereosinophilia with esosinophilic gastrointestinal disease, asthma"
Documents eosinophilic gastrointestinal disease as part of the phenotype.
Anaphylaxis Food-induced anaphylaxis HP:0500095 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Food-induced anaphylaxis (HP:0500095). HP:0500095 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."
Documents anaphylaxis, in the context of IgE-mediated food allergy.
Cerebral aneurysm Dilatation of the cerebral artery HP:0004944 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Cerebral aneurysm, annotated with Dilatation of the cerebral artery (HP:0004944). HP:0004944 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"Cerebral aneurysm: reported in one patient in adulthood; may be fatal"
Documents a reported, potentially fatal cerebral aneurysm in STAT6 GOF disease.
Allergic rhinitis HP:0003193 Human Phenotype Ontology (HP) Relation: this clinical feature is this phenotype This clinical feature is Allergic rhinitis (HP:0003193). HP:0003193 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"rhinoconjunctivitis, multiple food allergies, drug allergies, eosinophilic"
Documents allergic rhinoconjunctivitis among the key atopic diagnostic factors.
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Genetic Associations

1
STAT6 (autosomal dominant causal gain-of-function variant)
Gene: STAT6 hgnc:11368 HUGO Gene Nomenclature Committee (hgnc) Relation: this disease-associated gene is this gene This disease-associated gene is STAT6 (hgnc:11368). hgnc:11368 is a gene from the HUGO Gene Nomenclature Committee.
Show evidence (3 references)
PMID:36884218 SUPPORT Human Clinical
"This study identifies heterozygous GOF variants in STAT6 as a novel autosomal dominant allergic disorder."
Establishes STAT6 heterozygous GOF variants as the cause of a novel autosomal dominant allergic disorder.
PMID:37316763 SUPPORT Human Clinical
"We identified a novel heterozygous germline mutation STAT6 c.1255G > C, p.D419H leading to overactivity of IL-4 JAK/STAT signalling pathway, in a kindred affected by early-onset atopic dermatitis, food allergy, eosinophilic asthma, anaphylaxis and follicular lymphoma."
Independent kindred confirming a recurrent DNA-binding-domain variant (p.D419H) as a germline GOF cause of the disease.
PMID:40502541 SUPPORT Human Clinical
"This case report presents a new genetic variant that causes STAT6 gain-of-function disease in 2 patients, expands the clinical phenotype of STAT6 gain-of-function disease"
Independent report of an additional disease-causing variant (p.D519N), broadening the allelic spectrum.
💊

Medical Actions

3
Dupilumab
Action: PharmacotherapyNCI Thesaurus (NCIT) Relation: this treatment is this clinical intervention This treatment is Pharmacotherapy (NCIT:C15986). NCIT:C15986 is a clinical intervention from the NCI Thesaurus. NCIT:C15986
Agent: dupilumab NCIT:C162455 NCI Thesaurus (NCIT) Relation: this treatment uses this therapeutic agent This treatment uses dupilumab (NCIT:C162455). NCIT:C162455 is a therapeutic agent from the NCI Thesaurus.
The anti-IL-4Ra monoclonal antibody dupilumab blocks IL-4/IL-13 signaling upstream of STAT6 and was highly effective in STAT6 GOF disease, improving both clinical manifestations and immunological biomarkers.
Mechanism Target:
INHIBITS Constitutive STAT6 signaling — Blocking the shared IL-4Ra chain reduces IL-4/IL-13-driven input into the hyperresponsive STAT6 pathway.
Show evidence (2 references)
PMID:36884218 SUPPORT Human Clinical
"Precision treatment with the anti-IL-4Rα antibody, dupilumab, was highly effective improving both clinical manifestations and immunological biomarkers."
Documents dupilumab as an effective precision therapy.
PMID:40502541 SUPPORT Human Clinical
"p.D519N is a new disease-causing variant that responds well to dupilumab treatment"
Independent report of a successful dupilumab response in STAT6 GOF disease (p.D519N).
JAK inhibitor (ruxolitinib or tofacitinib)
Action: PharmacotherapyNCI Thesaurus (NCIT) Relation: this treatment is this clinical intervention This treatment is Pharmacotherapy (NCIT:C15986). NCIT:C15986 is a clinical intervention from the NCI Thesaurus. NCIT:C15986
Agent: ruxolitinib CHEBI:66919 Chemical Entities of Biological Interest (CHEBI) Relation: this treatment uses this therapeutic agent This treatment uses ruxolitinib (CHEBI:66919). CHEBI:66919 is a therapeutic agent from Chemical Entities of Biological Interest. tofacitinib CHEBI:71200 Chemical Entities of Biological Interest (CHEBI) Relation: this treatment uses this therapeutic agent This treatment uses tofacitinib (CHEBI:71200). CHEBI:71200 is a therapeutic agent from Chemical Entities of Biological Interest.
JAK inhibition targets the kinases upstream of STAT6. Ruxolitinib reversed STAT6 hyperresponsiveness to IL-4, normalized TH1/TH17 cells, suppressed eosinophilia, and improved atopic dermatitis; the consortium review names both ruxolitinib and tofacitinib as JAK inhibitors used in patients.
Mechanism Target:
INHIBITS Constitutive STAT6 signaling — JAK1/2 inhibition blocks the kinases upstream of STAT6, reducing STAT6 phosphorylation and downstream type 2 signaling.
Show evidence (3 references)
PMID:38238227 SUPPORT Human Clinical
"JAK inhibitors (ruxolitinib or tofacitinib)"
The consortium review names both ruxolitinib and tofacitinib as JAK inhibitors used in STAT6 GOF disease.
PMID:36758835 SUPPORT Human Clinical
"Treatment with the Janus kinase 1/2 inhibitor ruxolitinib reversed STAT6 hyperresponsiveness to IL-4, normalized TH1 and TH17 cells, suppressed the eosinophilia, and improved the patient's atopic dermatitis."
Documents ruxolitinib efficacy targeting the STAT6 signaling axis.
PMID:37316763 SUPPORT In Vitro
"The selective JAK1/JAK2 inhibitor ruxolitinib reduced pSTAT6 levels in D419H HEK293T cells and patient PBMC."
Pharmacodynamic evidence that ruxolitinib lowers pathological STAT6 phosphorylation in a patient-derived GOF variant.
Supportive and anaphylaxis-preparedness care
Action: supportive careNCI Thesaurus (NCIT) Relation: this treatment is this clinical intervention This treatment is supportive care (NCIT:C15747). NCIT:C15747 is a clinical intervention from the NCI Thesaurus. Ontology label: Supportive Care NCIT:C15747
Supportive management including allergen avoidance in sensitized patients, epinephrine autoinjectors and medical-alert measures for anaphylaxis, and bone-loss prophylaxis in patients on chronic corticosteroids. Anaphylaxis was fatal in one of the two reported deaths, underscoring the need for anaphylaxis preparedness.
Target Phenotypes: Food-induced anaphylaxis HP:0500095 Human Phenotype Ontology (HP) Relation: this treatment targets this phenotype This treatment targets Food-induced anaphylaxis (HP:0500095). HP:0500095 is a phenotype from the Human Phenotype Ontology.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"alert jewelry, epinephrine autoinjectors; immunization; prophylaxis for bone"
The consortium review specifies epinephrine autoinjectors, medical-alert measures, and bone-loss prophylaxis as supportive management.
🔬

Biochemical Markers

3
Serum IgE (INCREASED)
Context: Markedly elevated serum IgE reflects STAT6-driven IgE class switching.
Pathograph Readouts
Readout Of IgE class switching Positive Diagnostic
Elevated IgE reports the type 2 / IgE class-switching effector arm.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."
Elevated serum IgE is a diagnostic readout of the disease.
Show evidence (1 reference)
PMID:36884218 SUPPORT Human Clinical
"asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."
Documents elevated serum IgE as a biochemical hallmark.
Blood eosinophil count (INCREASED)
Context: Hypereosinophilia is a characteristic laboratory finding.
Pathograph Readouts
Readout Of Eosinophil expansion Positive Diagnostic
Blood eosinophilia reports the eosinophil effector arm of the type 2 response.
Show evidence (1 reference)
PMID:36758835 SUPPORT Human Clinical
"who presented with severe atopic dermatitis, eosinophilia, and elevated IgE."
Eosinophilia is a diagnostic readout in affected patients.
Pharmacodynamic Marker Of Eosinophil expansion Positive Pharmacodynamic
Eosinophil count is a pharmacodynamic marker of the eosinophil effector arm: it falls with dupilumab or JAK-inhibitor therapy and may track treatment efficacy.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"eosinophil count tends to be reduced after dupilumab or"
Eosinophil count decreases after dupilumab or JAK-inhibitor therapy, supporting a treatment-response readout.
Show evidence (1 reference)
PMID:36758835 SUPPORT Human Clinical
"who presented with severe atopic dermatitis, eosinophilia, and elevated IgE."
Documents eosinophilia as a biochemical hallmark.
Serum CCL24 (eotaxin-2) (INCREASED)
Context: The STAT6-regulated eosinophil chemokine CCL24 / eotaxin-2 is elevated in the serum of patients with STAT6 GOF disease, consistent with the eosinophil effector arm.
Pathograph Readouts
Readout Of Eosinophil expansion Positive Diagnostic
Elevated serum CCL24/eotaxin-2 reports STAT6-driven eosinophil chemotaxis.
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"was higher in s era from patients with STAT6 GOF and in gastric"
The STAT6-regulated chemokine CCL24/eotaxin-2 is elevated in patient sera (snippet preserves the source PDF's "s era" extraction artifact).
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"chemokine C-C motif chemokine ligand 24 [CCL24"
Identifies CCL24 (eotaxin-2) as a STAT6-regulated eosinophil chemokine relevant to the disease.
🔬

Diagnosis

4
Next-generation genetic sequencing
Molecular confirmation of a heterozygous STAT6 GOF variant establishes the diagnosis; NGS is described as the most powerful and cost-effective approach.
molecular genetic testing NCIT:C19770 NCI Thesaurus (NCIT)
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"Next-generation genetic sequencing: most powerful and cost-effective"
NGS is the recommended definitive diagnostic test for STAT6 GOF disease.
Serum total IgE and blood eosinophil count
Supportive laboratory findings: markedly raised total IgE and elevated absolute eosinophil count, with generally normal lymphocyte subsets.
clinical assessment NCIT:C124351 NCI Thesaurus (NCIT)
Show evidence (3 references)
PMID:38238227 SUPPORT Human Clinical
"Total IgE: raised; may exceed upper limit of detection"
Markedly raised total IgE is a supportive laboratory finding.
PMID:38238227 SUPPORT Human Clinical
"Complete blood count with white cell differentials; absolute eosinophil count"
Elevated absolute eosinophil count on CBC is a supportive finding.
PMID:38238227 SUPPORT Human Clinical
"Lymphocyte subsets: usually normal"
Lymphocyte subsets are usually normal, distinguishing from other IEIs.
Esophagogastroduodenoscopy
Upper GI endoscopy with biopsy documents eosinophilic esophageal disease (trachealization and furrowing, mucosal erosions, polypoid lesions).
esophagogastroduodenoscopy NCIT:C78144 NCI Thesaurus (NCIT)
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"erosions of mucosa, polypoid-like lesions; trachealization and furrowing in"
Upper GI endoscopy documents the eosinophilic esophageal disease component.
Colonoscopy
Lower GI endoscopy with biopsy documents eosinophilic intestinal disease (nodularities and lymphonodular hyperplasia).
colonoscopy NCIT:C16450 NCI Thesaurus (NCIT)
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"nodularities and lymphonodular hyperplasia in small and large"
Lower GI endoscopy documents the eosinophilic intestinal disease component.
📈

Progression

1
Prognosis is variable; most patients are managed with type 2-directed or JAK inhibitor therapy. Serious complications include lymphoma, kidney failure, and cerebral aneurysm. Two of 21 reported patients have died — from a cerebral aneurysm (age 35) and anaphylaxis (age 20).
Show evidence (2 references)
PMID:38238227 SUPPORT Human Clinical
"two patients out of 21 reported to date have died: causes were"
Documents disease-associated mortality (2 of 21 reported patients).
PMID:38238227 SUPPORT Human Clinical
"cerebral aneurysm (age 35 years) and anaphylaxis (age 20 years)"
Specifies the two fatal complications and ages at death.
📊

Prevalence

1
Worldwide (reported cohorts)
Cases In Literature Ultra Rare
Newly described entity; 21 individuals from 13 distinct families reported to date (as of the 2024 consortium review).
Show evidence (1 reference)
PMID:38238227 SUPPORT Human Clinical
"21 individuals from 13 distinct families have been"
Quantifies the cases-in-literature count for this newly described disease.
{ }

Source YAML

click to show
name: STAT6 Gain-of-Function Disease
creation_date: "2026-07-29T00:00:00Z"
category: Mendelian
description: >-
  STAT6 gain-of-function (GOF) disease is a recently described autosomal
  dominant inborn error of immunity caused by germline heterozygous
  gain-of-function variants in STAT6, the transcription factor downstream of the
  type 2 cytokines IL-4 and IL-13. GOF variants (predominantly in the DNA-binding
  domain) cause constitutive/hyperresponsive STAT6 signaling with sustained
  phosphorylation, increased target-gene expression, and TH2 skewing, producing a
  profound early-life multisystem allergic phenotype: treatment-resistant atopic
  dermatitis, marked hypereosinophilia with eosinophilic gastrointestinal
  disease, asthma, very high serum IgE, IgE-mediated food allergy, and
  anaphylaxis, with variable susceptibility to infection. It is catalogued in
  OMIM as hyper-IgE syndrome 6 (HIES6). Type 2-directed therapy (the anti-IL-4Ra
  antibody dupilumab) and JAK inhibition (ruxolitinib) are effective targeted
  treatments.
disease_term:
  preferred_term: STAT6 gain-of-function disease
  term:
    id: MONDO:0957807
    label: hyper-IgE syndrome 6, autosomal dominant, with recurrent infections
synonyms:
- STAT6-GOF
- STAT6 GOF disease
- Hyper-IgE syndrome 6
- HIES6
- Autosomal dominant allergic disorder due to STAT6 gain-of-function
- Early-onset multisystem allergic disease with STAT6 gain-of-function
parents:
- hereditary disease
- inborn error of immunity
- hyper-IgE syndrome
inheritance:
- name: Autosomal dominant inheritance
  inheritance_term:
    preferred_term: Autosomal dominant inheritance
    term:
      id: HP:0000006
      label: Autosomal dominant inheritance
  penetrance: COMPLETE
  expressivity: VARIABLE
  description: >-
    STAT6 GOF disease follows an autosomal dominant inheritance pattern from
    monoallelic (heterozygous) STAT6 variants; cases are either de novo/sporadic
    or transmitted through affected kindreds. Penetrance is complete, with
    variable expressivity.
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      The cases were either sporadic (seven kindreds) or followed an autosomal
      dominant inheritance pattern (three kindreds).
    explanation: >-
      Documents both sporadic/de novo and autosomal dominant transmission of
      heterozygous STAT6 GOF variants across the discovery cohort.
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      STAT6-GOF disease demonstrated complete penetrance, although some clinical
      variability
    explanation: >-
      The consortium review reports complete penetrance with clinical
      variability (variable expressivity).
pathophysiology:
- name: STAT6 gain-of-function variant
  biological_scale: MOLECULAR
  description: >-
    Germline heterozygous rare variants in STAT6 (most in the DNA-binding
    domain, e.g. p.E372K, p.E377K) confer a gain of function: the mutant
    transcription factor shows increased DNA-binding affinity, a strong
    preference for nuclear localization, and spontaneous transcriptional
    activity.
  genes:
  - preferred_term: STAT6
    term:
      id: hgnc:11368
      label: STAT6
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      All patients carried monoallelic rare variants in STAT6 and functional
      studies established their gain-of-function (GOF) phenotype with sustained
      STAT6 phosphorylation, increased STAT6 target gene expression, and TH2
      skewing.
    explanation: >-
      Establishes monoallelic STAT6 variants with a functionally validated
      gain-of-function phenotype as the causal lesion.
  - reference: PMID:36216080
    reference_title: "A germline STAT6 gain-of-function variant is associated with early-onset allergies."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      We identified a heterozygous missense variant (c.1129G>A;p.Glu377Lys) in
      the DNA binding domain of STAT6 that was de novo in the index patient's
      father and was inherited by 2 of his 3 children.
    explanation: >-
      Localizes a representative GOF variant to the STAT6 DNA-binding domain.
  downstream:
  - target: Constitutive STAT6 signaling
    description: >-
      GOF variants drive sustained/spontaneous STAT6 pathway activation
      independent of, and hyperresponsive to, upstream IL-4/IL-13 cytokine input.
    causal_link_type: DIRECT
    evidence:
    - reference: PMID:36216080
      reference_title: "A germline STAT6 gain-of-function variant is associated with early-onset allergies."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        A germline STAT6 gain-of-function variant results in spontaneous
        activation of the STAT6 signaling pathway and is associated with an
        early-onset and severe allergic phenotype in humans.
      explanation: >-
        Links the GOF variant directly to spontaneous activation of STAT6
        signaling.
- name: Constitutive STAT6 signaling
  conforms_to: "jak_stat_pathway_activation#Constitutive STAT Activation and Nuclear Translocation"
  biological_scale: MOLECULAR
  description: >-
    STAT6 is the central transcription factor of the type 2 cytokine (IL-4/IL-13)
    response. GOF variants produce sustained basal and cytokine-induced STAT6
    phosphorylation and increased target-gene transcription, amplifying the
    allergic-inflammation program.
  biological_processes:
  - preferred_term: interleukin-4-mediated signaling pathway
    term:
      id: GO:0035771
      label: interleukin-4-mediated signaling pathway
    modifier: INCREASED
  - preferred_term: JAK-STAT signaling
    term:
      id: GO:0007259
      label: cell surface receptor signaling pathway via JAK-STAT
    modifier: INCREASED
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      STAT6 (signal transducer and activator of transcription 6) is a
      transcription factor that plays a central role in the pathophysiology of
      allergic inflammation.
    explanation: >-
      Establishes STAT6 as the central signaling node whose constitutive
      activity drives the disease.
  - reference: PMID:36758835
    reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
    supports: SUPPORT
    evidence_source: IN_VITRO
    snippet: >-
      The mutation augmented both basal and cytokine-induced STAT6
      phosphorylation without affecting dephosphorylation kinetics.
    explanation: >-
      Functional assay of the mutated STAT6 protein documents increased basal and
      cytokine-induced STAT6 phosphorylation as the proximal signaling
      abnormality.
  - reference: PMID:40603028
    reference_title: "[Mechanism of pathogenesis by a gain-of-function variant of STAT6 causing severe allergic diseases and potential for development of molecularly targeted drugs]."
    supports: SUPPORT
    evidence_source: IN_VITRO
    snippet: >-
      even in the absence of IL-4 stimulation, we observed the translocation of
      mutant STAT6 in its unphosphorylated state, which activated gene
      expression.
    explanation: >-
      Documents ligand- and phosphorylation-independent nuclear translocation of
      the D419N mutant, the most constitutive form of the signaling defect.
  - reference: PMID:40603028
    reference_title: "[Mechanism of pathogenesis by a gain-of-function variant of STAT6 causing severe allergic diseases and potential for development of molecularly targeted drugs]."
    supports: SUPPORT
    evidence_source: MODEL_ORGANISM
    snippet: >-
      Mutant STAT6 knock-in mice elicited an abnormal TH2-dominant immune
      response in vivo, with findings similar to those observed in patients.
    explanation: >-
      A patient-derived D419N knock-in mouse recapitulates the human TH2/allergic
      phenotype, validating the causal mechanism in vivo.
  - reference: PMID:28653395
    reference_title: "Poly-ADP ribose polymerase-14 limits severity of allergic skin disease."
    supports: SUPPORT
    evidence_source: MODEL_ORGANISM
    snippet: >-
      mice that express constitutively active Stat6 in T cells (Stat6VT) and
      develop spontaneous inflammation of the skin
    explanation: >-
      An independent constitutively active STAT6 mouse model (Stat6VT) develops
      spontaneous allergic skin inflammation, corroborating that constitutive
      STAT6 activity drives atopic disease.
  downstream:
  - target: TH2 immune skewing
    description: >-
      Hyperactive STAT6 signaling skews CD4+ T-cell differentiation toward the
      TH2 program while suppressing TH1 and TH17 responses.
    causal_link_type: DIRECT
    evidence:
    - reference: PMID:36758835
      reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        Naive lymphocytes from the affected patient displayed increased TH2- and
        suppressed TH1- and TH17-cell responses.
      explanation: >-
        Links constitutive STAT6 activity to TH2 skewing with reciprocal TH1/TH17
        suppression.
  - target: B-cell lymphoma predisposition
    description: >-
      Constitutive STAT6 activity is oncogenic in the B-cell lineage: the same
      DNA-binding-domain residues mutated in the germline (notably D419) are
      recurrently mutated somatically in follicular lymphoma, predisposing to
      B-cell lymphomagenesis.
    causal_link_type: INDIRECT_UNKNOWN_INTERMEDIATES
    evidence:
    - reference: PMID:38238227
      reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        STAT6 is frequently and recurrently mutated in follicular lymphomas and
        other B cell lymphomas
      explanation: >-
        The shared STAT6 mutational spectrum between germline GOF disease and
        somatic follicular lymphoma links constitutive STAT6 activity to
        lymphomagenesis.
- name: TH2 immune skewing
  biological_scale: CELLULAR
  description: >-
    Constitutive STAT6 activity biases naive CD4+ T cells toward TH2
    differentiation with elevated peripheral TH2 lymphocytes, producing the IL-4/
    IL-5/IL-13-dominated milieu that underlies allergic effector disease.
  cell_types:
  - preferred_term: T-helper 2 cell
    term:
      id: CL:0000546
      label: T-helper 2 cell
  biological_processes:
  - preferred_term: T-helper 2 cell differentiation
    term:
      id: GO:0045064
      label: T-helper 2 cell differentiation
    modifier: INCREASED
  evidence:
  - reference: PMID:36216080
    reference_title: "A germline STAT6 gain-of-function variant is associated with early-onset allergies."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: Higher levels of peripheral blood TH2 lymphocytes were detected.
    explanation: >-
      Documents increased peripheral TH2 lymphocytes as the cellular readout of
      STAT6-driven skewing.
  downstream:
  - target: IgE class switching
    description: >-
      TH2 cytokines (IL-4/IL-13) drive B-cell immunoglobulin class switching to
      IgE, the humoral effector arm of the allergic phenotype.
    causal_link_type: DIRECT
  - target: Eosinophil expansion
    description: >-
      TH2 cytokines (IL-5) drive eosinophil expansion and tissue recruitment,
      the cellular effector arm of the allergic phenotype.
    causal_link_type: DIRECT
  - target: Impaired antimicrobial immunity
    description: >-
      Reciprocal suppression of TH1/TH17 responses contributes to recurrent and
      severe infection susceptibility in some patients.
    causal_link_type: INDIRECT_KNOWN_INTERMEDIATES
    intermediate_mechanisms:
    - TH1 response suppression
    - TH17 response suppression
    evidence:
    - reference: PMID:36758835
      reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        Naive lymphocytes from the affected patient displayed increased TH2- and
        suppressed TH1- and TH17-cell responses.
      explanation: >-
        TH1/TH17 suppression provides a mechanistic basis for impaired
        antimicrobial defense.
- name: IgE class switching
  biological_scale: CELLULAR
  description: >-
    The type 2 milieu drives B-cell immunoglobulin class switching to IgE,
    producing very high serum IgE — the humoral effector arm.
  cell_types:
  - preferred_term: B cell
    term:
      id: CL:0000236
      label: B cell
  biological_processes:
  - preferred_term: isotype switching to IgE isotypes
    term:
      id: GO:0035708
      label: interleukin-4-dependent isotype switching to IgE isotypes
    modifier: INCREASED
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      hypereosinophilia with esosinophilic gastrointestinal disease, asthma,
      elevated serum IgE, IgE-mediated food allergies, and anaphylaxis.
    explanation: >-
      Documents elevated serum IgE (and IgE-mediated food allergy) as the
      humoral effector consequence of the type 2 program.
  downstream:
  - target: Multisystem allergic disease
    description: >-
      IgE-mediated hypersensitivity drives food allergy, anaphylaxis, and atopic
      end-organ manifestations.
    causal_link_type: DIRECT
- name: Eosinophil expansion
  biological_scale: CELLULAR
  description: >-
    The type 2 milieu (IL-5) drives marked eosinophil expansion and tissue
    recruitment, producing blood hypereosinophilia and eosinophilic
    tissue infiltration — the cellular effector arm.
  cell_types:
  - preferred_term: eosinophil
    term:
      id: CL:0000771
      label: eosinophil
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      hypereosinophilia with esosinophilic gastrointestinal disease, asthma,
      elevated serum IgE, IgE-mediated food allergies, and anaphylaxis.
    explanation: >-
      Documents hypereosinophilia and eosinophilic gastrointestinal disease as
      the cellular effector consequence of the type 2 program.
  downstream:
  - target: Multisystem allergic disease
    description: >-
      Eosinophilic tissue infiltration drives eosinophilic gastrointestinal
      disease and other atopic end-organ manifestations.
    causal_link_type: DIRECT
- name: Multisystem allergic disease
  biological_scale: ORGANISM
  description: >-
    The convergent clinical endpoint: early-onset, treatment-resistant atopic
    dermatitis, asthma, eosinophilic gastrointestinal disease, IgE-mediated food
    allergy, and anaphylaxis.
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      a profound phenotype of early-life onset allergic immune dysregulation,
      widespread treatment-resistant atopic dermatitis, hypereosinophilia with
      esosinophilic gastrointestinal disease, asthma, elevated serum IgE,
      IgE-mediated food allergies, and anaphylaxis.
    explanation: >-
      Enumerates the multisystem allergic phenotype that defines the disease.
- name: Impaired antimicrobial immunity
  biological_scale: CELLULAR
  description: >-
    Reciprocal suppression of TH1 and TH17 responses (the mirror image of TH2
    skewing) impairs antimicrobial defense, underlying the recurrent skin,
    respiratory, and viral infections seen in a subset of patients and the OMIM
    designation of HIES6 as "with recurrent infections."
  cell_types:
  - preferred_term: T-helper 1 cell
    term:
      id: CL:0000545
      label: T-helper 1 cell
  - preferred_term: T-helper 17 cell
    term:
      id: CL:0000899
      label: T-helper 17 cell
  biological_processes:
  - preferred_term: T-helper 1 cell differentiation
    term:
      id: GO:0045063
      label: T-helper 1 cell differentiation
    modifier: DECREASED
  - preferred_term: T-helper 17 cell differentiation
    term:
      id: GO:0072539
      label: T-helper 17 cell differentiation
    modifier: DECREASED
  evidence:
  - reference: PMID:36758835
    reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Naive lymphocytes from the affected patient displayed increased TH2- and
      suppressed TH1- and TH17-cell responses.
    explanation: >-
      TH1/TH17 suppression provides the immunological basis for impaired
      antimicrobial defense.
  downstream:
  - target: Recurrent infections
    description: >-
      TH1/TH17 suppression manifests clinically as recurrent skin, respiratory,
      and viral infections.
    causal_link_type: DIRECT
    evidence:
    - reference: PMID:38238227
      reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        with recurrent skin, respiratory, and viral infections, but no fatal
        infections were noted.
      explanation: >-
        The consortium review documents recurrent skin, respiratory, and viral
        infections in a subset of patients.
- name: B-cell lymphoma predisposition
  biological_scale: CELLULAR
  description: >-
    STAT6 is a recurrently mutated oncogenic driver in follicular lymphoma and
    other B-cell lymphomas, and germline STAT6 GOF is associated with an emerging
    lymphoma risk: one reported patient developed follicular lymphoma that later
    relapsed as diffuse large B-cell lymphoma. The true magnitude of risk is not
    yet established.
  cell_types:
  - preferred_term: B cell
    term:
      id: CL:0000236
      label: B cell
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      To date, one patient found to have STAT6-GOF disease has developed
      lymphoma
    explanation: >-
      Documents the first reported lymphoma in a patient with germline STAT6 GOF
      disease.
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: OTHER
    snippet: >-
      STAT6 is frequently and recurrently mutated in follicular lymphomas and
      other B cell lymphomas
    explanation: >-
      Provides the biological rationale linking constitutive STAT6 activity to
      B-cell lymphomagenesis.
  - reference: PMID:37316763
    reference_title: "Autosomal Dominant STAT6 Gain of Function Causes Severe Atopy Associated with Lymphoma."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      The clinical association of lymphoma in our kindred, along with previous
      data linking somatic STAT6 D419H mutations to follicular lymphoma suggest
      that patients with STAT6 GOF disease may be at higher risk of
      lymphomagenesis.
    explanation: >-
      Independent kindred (germline p.D419H) directly linking STAT6 GOF disease
      to lymphoma risk, reinforcing the shared-residue rationale.
  downstream:
  - target: Lymphoma
    description: >-
      The lymphomagenic predisposition manifests clinically as B-cell lymphoma
      (follicular lymphoma, with reported transformation to diffuse large B-cell
      lymphoma).
    causal_link_type: INDIRECT_UNKNOWN_INTERMEDIATES
    evidence:
    - reference: PMID:38238227
      reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        a relapse with diffuse large B cell lymphoma at the age of 60 years
      explanation: >-
        Documents the follicular-to-DLBCL transformation in the index lymphoma
        case.
phenotypes:
- name: Atopic dermatitis
  category: Dermatological
  diagnostic: true
  description: >-
    Widespread, early-onset, treatment-resistant atopic dermatitis is the most
    consistent manifestation of STAT6 GOF disease.
  phenotype_term:
    preferred_term: Atopic dermatitis
    term:
      id: HP:0001047
      label: Atopic dermatitis
    onset:
      onset_category: INFANTILE
      notes: Disease onset in early infancy across the reported cohort.
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      a profound phenotype of early-life onset allergic immune dysregulation,
      widespread treatment-resistant atopic dermatitis
    explanation: Documents widespread treatment-resistant atopic dermatitis as a core feature.
- name: Increased circulating IgE concentration
  category: Immunological
  diagnostic: true
  description: >-
    Markedly elevated serum IgE is a hallmark laboratory feature, reflecting the
    STAT6-driven IgE class switching.
  phenotype_term:
    preferred_term: Increased circulating IgE concentration
    term:
      id: HP:0003212
      label: Increased circulating IgE concentration
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis.
    explanation: Documents elevated serum IgE as part of the core phenotype.
- name: Eosinophilia
  category: Immunological
  description: >-
    Marked blood hypereosinophilia is characteristic and can be accompanied by
    tissue eosinophilic infiltration.
  phenotype_term:
    preferred_term: Increased total eosinophil count
    term:
      id: HP:0001880
      label: Increased total eosinophil count
  evidence:
  - reference: PMID:36758835
    reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      who presented with severe atopic dermatitis, eosinophilia, and elevated
      IgE.
    explanation: Documents eosinophilia in an affected patient.
- name: Food allergy
  category: Immunological
  description: >-
    IgE-mediated food allergy is a key presentation and a source of
    life-threatening anaphylaxis.
  phenotype_term:
    preferred_term: Food allergy
    term:
      id: HP:0500093
      label: Food allergy
  evidence:
  - reference: PMID:36216080
    reference_title: "A germline STAT6 gain-of-function variant is associated with early-onset allergies."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: Severe atopic dermatitis and food allergy were key presentations.
    explanation: Documents food allergy as a key presentation.
- name: Asthma
  category: Respiratory
  description: Asthma is part of the multisystem atopic phenotype.
  phenotype_term:
    preferred_term: Asthma
    term:
      id: HP:0002099
      label: Asthma
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      hypereosinophilia with esosinophilic gastrointestinal disease, asthma,
      elevated serum IgE
    explanation: Documents asthma as part of the phenotype.
- name: Eosinophilic esophagitis
  category: Gastrointestinal
  description: >-
    Eosinophilic gastrointestinal disease, including eosinophilic esophagitis, is
    part of the STAT6 GOF phenotype.
  phenotype_term:
    preferred_term: Eosinophilic esophagitis
    term:
      id: HP:0410151
      label: Eosinophilic infiltration of the esophagus
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: hypereosinophilia with esosinophilic gastrointestinal disease, asthma
    explanation: Documents eosinophilic gastrointestinal disease as part of the phenotype.
- name: Anaphylaxis
  category: Immunological
  description: >-
    IgE-mediated anaphylaxis, frequently food-induced, occurs in STAT6 GOF
    disease.
  phenotype_term:
    preferred_term: Food-induced anaphylaxis
    term:
      id: HP:0500095
      label: Food-induced anaphylaxis
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: elevated serum IgE, IgE-mediated food allergies, and anaphylaxis.
    explanation: Documents anaphylaxis, in the context of IgE-mediated food allergy.
- name: Recurrent infections
  category: Immunological
  description: >-
    A subset of patients has increased susceptibility to recurrent infection,
    consistent with the OMIM designation as a hyper-IgE syndrome with recurrent
    infections and with reciprocal TH1/TH17 suppression.
  phenotype_term:
    preferred_term: Recurrent infections
    term:
      id: HP:0002719
      label: Recurrent infections
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      with recurrent skin, respiratory, and viral infections, but no fatal
      infections were noted.
    explanation: >-
      The consortium review documents recurrent skin, respiratory, and viral
      infections in a subset of patients.
  - reference: PMID:36758835
    reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Naive lymphocytes from the affected patient displayed increased TH2- and
      suppressed TH1- and TH17-cell responses.
    explanation: >-
      TH1/TH17 suppression provides an immunological basis for infection
      susceptibility; recurrent infection is captured in the OMIM disease name.
- name: Lymphoma
  category: Oncologic
  description: >-
    Germline STAT6 GOF carries an emerging predisposition to B-cell lymphoma;
    the first reported case developed follicular lymphoma that later relapsed as
    diffuse large B-cell lymphoma. True lifetime risk is not yet established.
  phenotype_term:
    preferred_term: B-cell lymphoma
    term:
      id: HP:0002665
      label: Lymphoma
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      To date, one patient found to have STAT6-GOF disease has developed
      lymphoma
    explanation: >-
      Documents the first reported lymphoma in a patient with germline STAT6 GOF
      disease.
- name: Cerebral aneurysm
  category: Neurologic
  description: >-
    A cerebral aneurysm has been reported as a non-immunological feature (in the
    spectrum shared with STAT3-related HIES) and was fatal in one patient; the
    causal relationship to the STAT6 GOF variant is not yet established.
  phenotype_term:
    preferred_term: Cerebral aneurysm
    term:
      id: HP:0004944
      label: Dilatation of the cerebral artery
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Cerebral aneurysm: reported in one patient in adulthood; may be fatal
    explanation: >-
      Documents a reported, potentially fatal cerebral aneurysm in STAT6 GOF
      disease.
- name: Short stature
  category: Growth
  description: >-
    Short stature is reported as a non-immunological feature overlapping the
    STAT3-LOF HIES spectrum.
  phenotype_term:
    preferred_term: Short stature
    term:
      id: HP:0004322
      label: Short stature
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      including short stature, pathological fractures,
    explanation: >-
      Documents short stature among the STAT3-LOF-overlapping non-immunological
      features of STAT6 GOF disease.
- name: Osteoporosis
  category: Musculoskeletal
  description: >-
    Osteoporosis with pathological fractures is reported as a non-immunological
    feature of STAT6 GOF disease.
  phenotype_term:
    preferred_term: Osteoporosis with pathological fractures
    term:
      id: HP:0000939
      label: Osteoporosis
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      osteoporosis with pathological fractures, generalized joint
    explanation: >-
      Documents osteoporosis with pathological fractures as a reported feature.
- name: Gastroesophageal reflux
  category: Gastrointestinal
  description: >-
    Early gastroesophageal reflux disease is part of the gastrointestinal
    manifestations.
  phenotype_term:
    preferred_term: Gastroesophageal reflux
    term:
      id: HP:0002020
      label: Gastroesophageal reflux
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      gastroesophageal reflux disease
    explanation: >-
      Documents early gastroesophageal reflux disease as a diagnostic feature.
- name: Allergic rhinitis
  category: Immunological
  description: >-
    Allergic rhinitis (part of allergic rhinoconjunctivitis) is part of the
    multisystem atopic phenotype.
  phenotype_term:
    preferred_term: Allergic rhinitis
    term:
      id: HP:0003193
      label: Allergic rhinitis
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      rhinoconjunctivitis, multiple food allergies, drug allergies, eosinophilic
    explanation: >-
      Documents allergic rhinoconjunctivitis among the key atopic diagnostic
      factors.
- name: Lymphadenopathy
  category: Immunological
  description: >-
    Lymphadenopathy is a feature of the lymphoproliferation seen in STAT6 GOF
    disease.
  phenotype_term:
    preferred_term: Lymphadenopathy
    term:
      id: HP:0002716
      label: Lymphadenopathy
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Lymphoproliferation, characterized by lymphadenopathy
    explanation: >-
      Documents lymphadenopathy as a feature of STAT6 GOF lymphoproliferation.
biochemical:
- name: Serum IgE
  presence: INCREASED
  context: Markedly elevated serum IgE reflects STAT6-driven IgE class switching.
  biomarker_term:
    preferred_term: Increased circulating IgE concentration
    term:
      id: HP:0003212
      label: Increased circulating IgE concentration
  readouts:
  - target: IgE class switching
    relationship: READOUT_OF
    direction: POSITIVE
    endpoint_context: DIAGNOSTIC
    interpretation: Elevated IgE reports the type 2 / IgE class-switching effector arm.
    evidence:
    - reference: PMID:36884218
      reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis.
      explanation: Elevated serum IgE is a diagnostic readout of the disease.
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis.
    explanation: Documents elevated serum IgE as a biochemical hallmark.
- name: Blood eosinophil count
  presence: INCREASED
  context: Hypereosinophilia is a characteristic laboratory finding.
  biomarker_term:
    preferred_term: Increased total eosinophil count
    term:
      id: HP:0001880
      label: Increased total eosinophil count
  readouts:
  - target: Eosinophil expansion
    relationship: READOUT_OF
    direction: POSITIVE
    endpoint_context: DIAGNOSTIC
    interpretation: Blood eosinophilia reports the eosinophil effector arm of the type 2 response.
    evidence:
    - reference: PMID:36758835
      reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: who presented with severe atopic dermatitis, eosinophilia, and elevated IgE.
      explanation: Eosinophilia is a diagnostic readout in affected patients.
  - target: Eosinophil expansion
    relationship: PHARMACODYNAMIC_MARKER_OF
    direction: POSITIVE
    endpoint_context: PHARMACODYNAMIC
    interpretation: >-
      Eosinophil count is a pharmacodynamic marker of the eosinophil effector
      arm: it falls with dupilumab or JAK-inhibitor therapy and may track
      treatment efficacy.
    evidence:
    - reference: PMID:38238227
      reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        eosinophil count tends to be reduced after dupilumab or
      explanation: >-
        Eosinophil count decreases after dupilumab or JAK-inhibitor therapy,
        supporting a treatment-response readout.
  evidence:
  - reference: PMID:36758835
    reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: who presented with severe atopic dermatitis, eosinophilia, and elevated IgE.
    explanation: Documents eosinophilia as a biochemical hallmark.
- name: Serum CCL24 (eotaxin-2)
  presence: INCREASED
  context: >-
    The STAT6-regulated eosinophil chemokine CCL24 / eotaxin-2 is elevated in
    the serum of patients with STAT6 GOF disease, consistent with the eosinophil
    effector arm.
  biomarker_term:
    preferred_term: C-C motif chemokine 24 (eotaxin-2)
    term:
      id: NCIT:C28736
      label: C-C Motif Chemokine 24
  readouts:
  - target: Eosinophil expansion
    relationship: READOUT_OF
    direction: POSITIVE
    endpoint_context: DIAGNOSTIC
    interpretation: >-
      Elevated serum CCL24/eotaxin-2 reports STAT6-driven eosinophil chemotaxis.
    evidence:
    - reference: PMID:38238227
      reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        was higher in s era from patients with STAT6 GOF and in gastric
      explanation: >-
        The STAT6-regulated chemokine CCL24/eotaxin-2 is elevated in patient
        sera (snippet preserves the source PDF's "s era" extraction artifact).
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      chemokine C-C motif chemokine ligand 24 [CCL24
    explanation: >-
      Identifies CCL24 (eotaxin-2) as a STAT6-regulated eosinophil chemokine
      relevant to the disease.
genetic:
- name: STAT6
  gene_term:
    preferred_term: STAT6
    term:
      id: hgnc:11368
      label: STAT6
  association: autosomal dominant causal gain-of-function variant
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      This study identifies heterozygous GOF variants in STAT6 as a novel
      autosomal dominant allergic disorder.
    explanation: >-
      Establishes STAT6 heterozygous GOF variants as the cause of a novel
      autosomal dominant allergic disorder.
  - reference: PMID:37316763
    reference_title: "Autosomal Dominant STAT6 Gain of Function Causes Severe Atopy Associated with Lymphoma."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      We identified a novel heterozygous germline mutation STAT6 c.1255G > C,
      p.D419H leading to overactivity of IL-4 JAK/STAT signalling pathway, in a
      kindred affected by early-onset atopic dermatitis, food allergy,
      eosinophilic asthma, anaphylaxis and follicular lymphoma.
    explanation: >-
      Independent kindred confirming a recurrent DNA-binding-domain variant
      (p.D419H) as a germline GOF cause of the disease.
  - reference: PMID:40502541
    reference_title: "STAT6 gain-of-function disease: p.D519N is a new disease-causing variant that responds well to dupilumab treatment."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      This case report presents a new genetic variant that causes STAT6
      gain-of-function disease in 2 patients, expands the clinical phenotype of
      STAT6 gain-of-function disease
    explanation: >-
      Independent report of an additional disease-causing variant (p.D519N),
      broadening the allelic spectrum.
treatments:
- name: Dupilumab
  description: >-
    The anti-IL-4Ra monoclonal antibody dupilumab blocks IL-4/IL-13 signaling
    upstream of STAT6 and was highly effective in STAT6 GOF disease, improving
    both clinical manifestations and immunological biomarkers.
  therapeutic_modality: MONOCLONAL_ANTIBODY
  treatment_term:
    preferred_term: Pharmacotherapy
    term:
      id: NCIT:C15986
      label: Pharmacotherapy
    therapeutic_agent:
    - preferred_term: dupilumab
      term:
        id: NCIT:C162455
        label: Dupilumab
  evidence:
  - reference: PMID:36884218
    reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Precision treatment with the anti-IL-4Rα antibody, dupilumab, was highly
      effective improving both clinical manifestations and immunological
      biomarkers.
    explanation: Documents dupilumab as an effective precision therapy.
  - reference: PMID:40502541
    reference_title: "STAT6 gain-of-function disease: p.D519N is a new disease-causing variant that responds well to dupilumab treatment."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      p.D519N is a new disease-causing variant that responds well to dupilumab
      treatment
    explanation: >-
      Independent report of a successful dupilumab response in STAT6 GOF disease
      (p.D519N).
  target_mechanisms:
  - target: Constitutive STAT6 signaling
    treatment_effect: INHIBITS
    description: >-
      Blocking the shared IL-4Ra chain reduces IL-4/IL-13-driven input into the
      hyperresponsive STAT6 pathway.
- name: JAK inhibitor (ruxolitinib or tofacitinib)
  description: >-
    JAK inhibition targets the kinases upstream of STAT6. Ruxolitinib reversed
    STAT6 hyperresponsiveness to IL-4, normalized TH1/TH17 cells, suppressed
    eosinophilia, and improved atopic dermatitis; the consortium review names
    both ruxolitinib and tofacitinib as JAK inhibitors used in patients.
  therapeutic_modality: SMALL_MOLECULE
  treatment_term:
    preferred_term: Pharmacotherapy
    term:
      id: NCIT:C15986
      label: Pharmacotherapy
    therapeutic_agent:
    - preferred_term: ruxolitinib
      term:
        id: CHEBI:66919
        label: ruxolitinib
    - preferred_term: tofacitinib
      term:
        id: CHEBI:71200
        label: tofacitinib
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      JAK inhibitors (ruxolitinib or tofacitinib)
    explanation: >-
      The consortium review names both ruxolitinib and tofacitinib as JAK
      inhibitors used in STAT6 GOF disease.
  - reference: PMID:36758835
    reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Treatment with the Janus kinase 1/2 inhibitor ruxolitinib reversed STAT6
      hyperresponsiveness to IL-4, normalized TH1 and TH17 cells, suppressed the
      eosinophilia, and improved the patient's atopic dermatitis.
    explanation: Documents ruxolitinib efficacy targeting the STAT6 signaling axis.
  - reference: PMID:37316763
    reference_title: "Autosomal Dominant STAT6 Gain of Function Causes Severe Atopy Associated with Lymphoma."
    supports: SUPPORT
    evidence_source: IN_VITRO
    snippet: >-
      The selective JAK1/JAK2 inhibitor ruxolitinib reduced pSTAT6 levels in
      D419H HEK293T cells and patient PBMC.
    explanation: >-
      Pharmacodynamic evidence that ruxolitinib lowers pathological STAT6
      phosphorylation in a patient-derived GOF variant.
  target_mechanisms:
  - target: Constitutive STAT6 signaling
    treatment_effect: INHIBITS
    description: >-
      JAK1/2 inhibition blocks the kinases upstream of STAT6, reducing STAT6
      phosphorylation and downstream type 2 signaling.
- name: Supportive and anaphylaxis-preparedness care
  description: >-
    Supportive management including allergen avoidance in sensitized patients,
    epinephrine autoinjectors and medical-alert measures for anaphylaxis, and
    bone-loss prophylaxis in patients on chronic corticosteroids. Anaphylaxis
    was fatal in one of the two reported deaths, underscoring the need for
    anaphylaxis preparedness.
  therapeutic_modality: BEHAVIORAL
  treatment_term:
    preferred_term: supportive care
    term:
      id: NCIT:C15747
      label: Supportive Care
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      alert jewelry, epinephrine autoinjectors; immunization; prophylaxis for bone
    explanation: >-
      The consortium review specifies epinephrine autoinjectors, medical-alert
      measures, and bone-loss prophylaxis as supportive management.
  target_phenotypes:
  - preferred_term: Food-induced anaphylaxis
    term:
      id: HP:0500095
      label: Food-induced anaphylaxis
diagnosis:
- name: Next-generation genetic sequencing
  description: >-
    Molecular confirmation of a heterozygous STAT6 GOF variant establishes the
    diagnosis; NGS is described as the most powerful and cost-effective approach.
  diagnosis_term:
    preferred_term: molecular genetic testing
    term:
      id: NCIT:C19770
      label: Molecular Analysis
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Next-generation genetic sequencing: most powerful and cost-effective
    explanation: >-
      NGS is the recommended definitive diagnostic test for STAT6 GOF disease.
- name: Serum total IgE and blood eosinophil count
  description: >-
    Supportive laboratory findings: markedly raised total IgE and elevated
    absolute eosinophil count, with generally normal lymphocyte subsets.
  diagnosis_term:
    preferred_term: clinical assessment
    term:
      id: NCIT:C124351
      label: Clinical Evaluation
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Total IgE: raised; may exceed upper limit of detection
    explanation: >-
      Markedly raised total IgE is a supportive laboratory finding.
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Complete blood count with white cell differentials; absolute eosinophil count
    explanation: >-
      Elevated absolute eosinophil count on CBC is a supportive finding.
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      Lymphocyte subsets: usually normal
    explanation: >-
      Lymphocyte subsets are usually normal, distinguishing from other IEIs.
- name: Esophagogastroduodenoscopy
  description: >-
    Upper GI endoscopy with biopsy documents eosinophilic esophageal disease
    (trachealization and furrowing, mucosal erosions, polypoid lesions).
  diagnosis_term:
    preferred_term: esophagogastroduodenoscopy
    term:
      id: NCIT:C78144
      label: Esophagogastroduodenoscopy
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      erosions of mucosa, polypoid-like lesions; trachealization and furrowing in
    explanation: >-
      Upper GI endoscopy documents the eosinophilic esophageal disease component.
- name: Colonoscopy
  description: >-
    Lower GI endoscopy with biopsy documents eosinophilic intestinal disease
    (nodularities and lymphonodular hyperplasia).
  diagnosis_term:
    preferred_term: colonoscopy
    term:
      id: NCIT:C16450
      label: Colonoscopy
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      nodularities and lymphonodular hyperplasia in small and large
    explanation: >-
      Lower GI endoscopy documents the eosinophilic intestinal disease component.
prevalence:
- population: Worldwide (reported cohorts)
  measure_type: CASES_IN_LITERATURE
  prevalence_class: ULTRA_RARE
  notes: >-
    Newly described entity; 21 individuals from 13 distinct families reported to
    date (as of the 2024 consortium review).
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      21 individuals from 13 distinct families have been
    explanation: >-
      Quantifies the cases-in-literature count for this newly described disease.
progression:
- notes: >-
    Prognosis is variable; most patients are managed with type 2-directed or JAK
    inhibitor therapy. Serious complications include lymphoma, kidney failure,
    and cerebral aneurysm. Two of 21 reported patients have died — from a
    cerebral aneurysm (age 35) and anaphylaxis (age 20).
  evidence:
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      two patients out of 21 reported to date have died: causes were
    explanation: >-
      Documents disease-associated mortality (2 of 21 reported patients).
  - reference: PMID:38238227
    reference_title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: >-
      cerebral aneurysm (age 35 years) and anaphylaxis (age 20 years)
    explanation: >-
      Specifies the two fatal complications and ages at death.
classifications:
  harrisons_chapter:
  - classification_value: IMMUNE_RHEUMATOLOGIC
    evidence:
    - reference: PMID:36758835
      reference_title: "Severe allergic dysregulation due to a gain of function mutation in the transcription factor STAT6."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        This study identified a novel inborn error of immunity due to a STAT6
        gain-of-function mutation that gave rise to severe allergic
        dysregulation.
      explanation: >-
        Frames the disease as an inborn error of immunity manifesting as severe
        allergic (immune-dysregulation) disease, supporting placement in the
        immunology/rheumatology Part.
  - classification_value: GENETICS_ENVIRONMENT_DISEASE
    evidence:
    - reference: PMID:36884218
      reference_title: "Human germline heterozygous gain-of-function STAT6 variants cause severe allergic disease."
      supports: SUPPORT
      evidence_source: HUMAN_CLINICAL
      snippet: >-
        This study identifies heterozygous GOF variants in STAT6 as a novel
        autosomal dominant allergic disorder.
      explanation: >-
        A monogenic (autosomal dominant) germline disorder, supporting placement
        in the genetics Part.
  iuis_category:
    classification_value: combined immunodeficiency with syndromic features
    notes: >-
      Corrected from `immune dysregulation` (2026-08-20). The IUIS 2024 update
      places STAT6 GOF in Table 2, subtable 1 — combined immunodeficiencies
      with syndromic features — not Table 4. The earlier assignment read the
      disease's dominant allergic/type-2 dysregulation phenotype as a Table 4
      signal, but IUIS groups it with the hyper-IgE-like syndromic entities
      alongside dominant-negative STAT3, where an immune defect is inseparable
      from a broader syndromic presentation. The phenotype description is
      unchanged; only the table assignment is.
    evidence:
    - reference: PMID:41608114
      reference_title: "Human inborn errors of immunity: 2024 update on the classification from the International Union of Immunological Societies Expert Committee."
      supports: SUPPORT
      evidence_source: OTHER
      snippet: >-
        Combined immunodeficiencies with syndromic features: IKZF2 (dominant
        negative); GINS4, SLC19A1, SGPL1, FLT3L, ITPR3, RECQL4 (AR LOF); PTCRA
        (AR LOF/hypomorphic); SMAD3 (AD); and STAT6 (AD GOF)
      explanation: >-
        The IUIS Expert Committee's own enumeration of gene defects new since
        the 2022 update lists STAT6 (AD GOF) under "combined immunodeficiencies
        with syndromic features", which the same sentence identifies as Table 2,
        subtable 1.
references:
- reference: PMID:38238227
  title: "Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond."
notes: >-
  Initial curation from the founding STAT6 GOF disease literature (Sharma et al.
  JEM 2023; Baris et al. JACI 2023; Suratannon et al. JACI 2023) plus the STAT6
  GOF International Consortium review. Emphasizes the STAT6 GOF -> constitutive
  type 2 signaling -> TH2 skewing -> IgE/eosinophil effector -> multisystem
  allergic disease axis and the dupilumab / JAK-inhibitor targeted treatments.
datasets: []
📚

References & Deep Research

References

1
Human germline gain-of-function in STAT6: from severe allergic disease to lymphoma and beyond.
No top-level findings curated for this source.

Deep Research

1
OpenScientist
STAT6 Gain-of-Function Disease (Hyper-IgE Syndrome 6, HIES6): A Comprehensive Disease Characterization Report
openscientist-autonomous 10 citations 2026-07-29T22:47:56.771194

STAT6 Gain-of-Function Disease (Hyper-IgE Syndrome 6, HIES6): A Comprehensive Disease Characterization Report

Summary

STAT6 gain-of-function (GOF) disease is a rare, recently described (2023) autosomal-dominant primary atopic disorder (PAD)—one of a growing group of inborn errors of immunity (IEIs) in which a single germline gene defect produces severe, early-onset allergic disease. It is caused by germline heterozygous activating (gain-of-function) missense variants in STAT6 (Signal Transducer and Activator of Transcription 6; chromosome 12q13.3; HGNC:11364; NCBI Gene 6778; OMIM 601512). Pathogenic variants cluster in the DNA-binding domain, with a recurrent hotspot at codon Asp419 (D419H/Y/G/N) and additional recurrent variants including E372K, E377K, E382Q, and D519H/N. These variants produce constitutive and/or ligand-hypersensitive IL-4/IL-13–JAK–STAT6 signaling, with sustained STAT6 phosphorylation, enhanced nuclear translocation (in some cases even without phosphorylation), increased STAT6 target-gene expression, and pathological TH2 skewing of the adaptive immune system.

Clinically, the disease presents in infancy (100% of the founding cohort) with a profound, multi-system allergic phenotype: widespread treatment-resistant atopic dermatitis (94%), hypereosinophilia and markedly elevated serum IgE (94%), IgE-mediated food allergy (94%), asthma (69%), eosinophilic gastrointestinal disease (63%), and anaphylaxis (56%). Variable features include recurrent skin/respiratory/viral infections, short stature, osteoporosis, and a small but important risk of B-cell/follicular lymphoma (~6%), mechanistically linked to the same DNA-binding-domain residues that are recurrently mutated somatically in follicular lymphoma. The disorder is catalogued as OMIM #620532 ("Hyper-IgE syndrome 6, autosomal dominant, with recurrent infections; HIES6") and MONDO:0957807.

The disease is highly actionable: because the driver is a hyperactive, druggable signaling axis, pathway-targeted therapy is transformative. The anti–IL-4Rα monoclonal antibody dupilumab and JAK inhibitors (e.g., ruxolitinib) improve both clinical manifestations and immunological biomarkers. Diagnosis relies on exome/genome sequencing with functional confirmation of STAT6 hyperactivation. Two constitutively active mouse models (Stat6VT transgenic and patient-derived D419N knock-in) recapitulate the human TH2/allergic phenotype and validate the causal mechanism. This report synthesizes 9 confirmed findings drawn from 11 reviewed papers into a full disease knowledge-base entry organized along the 15 requested characteristic domains, followed by a mechanistic model, evidence base, limitations, and proposed follow-up actions.


Key Findings

Finding 1 — STAT6 GOF disease is a novel autosomal-dominant primary atopic disorder caused by germline heterozygous gain-of-function STAT6 variants

The defining evidence comes from a landmark international cohort of 16 patients from 10 families across three continents (Sharma et al., 2023). All patients carried monoallelic (heterozygous) rare variants in STAT6, and functional studies established a gain-of-function phenotype. As the authors state verbatim: "All patients carried monoallelic rare variants in STAT6 and functional studies established their gain-of-function (GOF) phenotype with sustained STAT6 phosphorylation, increased STAT6 target gene expression, and TH2 skewing" and "This study identifies heterozygous GOF variants in STAT6 as a novel autosomal dominant allergic disorder" (PMID: 36884218). Inheritance was sporadic (de novo) in 7 kindreds and autosomal dominant in 3 kindreds, consistent with a dominant, GOF (not loss-of-function/haploinsufficiency) mechanism.

Evidence source: human clinical/genetic (multi-family cohort with functional validation).

Finding 2 — Core clinical phenotype: early-onset treatment-resistant atopic dermatitis, hypereosinophilia, eosinophilic GI disease, asthma, elevated IgE, food allergy and anaphylaxis

The founding cohort described "a profound phenotype of early-life onset allergic immune dysregulation, widespread treatment-resistant atopic dermatitis, hypereosinophilia with esosinophilic gastrointestinal disease, asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis" (PMID: 36884218). This multi-system atopic constellation is the diagnostic signature and is independently replicated in single-case/kindred reports: Baris et al. (E372K), Suratannon/independent (E377K), Minskaia (D419H), and Samra (D519N) each describe severe atopic dermatitis, eosinophilia, elevated IgE, and food allergy.

Evidence source: human clinical.

Finding 3 — Recurrent pathogenic variants cluster in the STAT6 DNA-binding domain and cause constitutive/enhanced IL-4/JAK/STAT6 signaling

Reported germline missense variants include p.E372K (c.1114G>A), p.E377K (c.1129G>A), p.E382Q (c.1144G>C), p.D419H (c.1255G>C), p.D419Y (c.1255G>T), p.D419G (c.1256A>G), p.D419N (c.1255G>A), and p.D519H/N (c.1555G>C)—several within the DNA-binding domain (DBD). Direct quotes anchor the mechanism: - "a missense mutation in the DNA binding domain of STAT6 (c.1114G>A, p.E372K)" (PMID: 36758835). - "a novel heterozygous germline mutation STAT6 c.1255G > C, p.D419H leading to overactivity of IL-4 JAK/STAT signalling pathway" (PMID: 37316763). - Ligand independence was shown for D419N: "even in the absence of IL-4 stimulation, we observed the translocation of mutant STAT6 in its unphosphorylated state, which activated gene expression" (PMID: 40603028).

Thus, some variants confer hypersensitivity to IL-4 (elevated total/phospho-STAT6 at baseline and after IL-4, e.g., D419H) while others confer constitutive, phosphorylation-independent nuclear translocation and transcription (D419N).

Evidence source: human genetic + in vitro functional (HEK293T, patient PBMC, gastric organoids).

Finding 4 — Targeted therapy: dupilumab and JAK inhibitors are effective; disease is associated with follicular lymphoma risk

Because the disease is driven by a hyperactive IL-4/IL-13–JAK–STAT6 axis, blocking that axis is therapeutic. "Precision treatment with the anti-IL-4Rα antibody, dupilumab, was highly effective improving both clinical manifestations and immunological biomarkers" (PMID: 36884218); dupilumab was also effective for the D519N variant (Samra 2025, PMID: 40502541). JAK inhibition targets the upstream kinases: "The selective JAK1/JAK2 inhibitor ruxolitinib reduced pSTAT6 levels in D419H HEK293T cells and patient PBMC" (PMID: 37316763). Critically, the same Minskaia kindred (D419H) included follicular lymphoma, linking germline STAT6 GOF to lymphomagenesis.

Evidence source: human clinical (treatment response) + in vitro (pharmacodynamic).

Finding 5 — Nosology and identifiers: OMIM #620532 (HIES6) / MONDO:0957807

STAT6 GOF disease is catalogued as OMIM #620532 = "HYPER-IgE SYNDROME 6, AUTOSOMAL DOMINANT, WITH RECURRENT INFECTIONS; HIES6." The Mondo term MONDO:0957807 ("hyper-IgE syndrome 6, autosomal dominant, with recurrent infections") cross-references OMIM:620532, GARD:0026874, MedGen:1851769, and UMLS:C5848786. The causal gene STAT6 = OMIM 601512, HGNC:11364, NCBI Gene 6778, UniProt P42226. NCI Thesaurus C212086 = "Activating STAT6 Gene Mutation." No dedicated Orphanet/ORDO code was identified at the time of research.

Evidence source: aggregated disease-level resources (OMIM, Mondo, MedGen, NCIt).

Finding 6 — Quantitative phenotype frequencies (HPO annotations, n=16 founding cohort)

Official HPO disease annotations (OMIM:620532 / MONDO:0957807), all sourced to PMID: 36884218, provide curated frequencies (see the phenotype table in Section 3). They derive from the cohort description: "widespread treatment-resistant atopic dermatitis, hypereosinophilia with esosinophilic gastrointestinal disease, asthma, elevated serum IgE, IgE-mediated food allergies, and anaphylaxis."

Evidence source: curated ontology annotation of human clinical cohort.

Finding 7 — ClinVar variant spectrum and gnomAD constraint support a DBD missense GOF mechanism (not haploinsufficiency)

ClinVar (transcript NM_003153.5) lists germline Pathogenic/Likely-pathogenic STAT6 variants for "Hyper-IgE syndrome 6": c.1114G>A p.Glu372Lys (P), c.1144G>C p.Glu382Gln (P), c.1255G>C p.Asp419His (LP), c.1255G>T p.Asp419Tyr (P), c.1256A>G p.Asp419Gly (P), and c.1555G>C p.Asp519His (P). Codon 419 is a recurrent hotspot. gnomAD constraint metrics show STAT6 is LoF-tolerant (pLI = 0.057; oe_lof upper bound = 0.54) but missense-constrained (mis_z = 3.47). This constraint signature—tolerant of loss-of-function but intolerant of missense change, combined with recurrent, clustered, dominant missense variants—is the classic fingerprint of a gain-of-function, not haploinsufficiency, disease mechanism.

Evidence source: population genomics / variant databases (computational).

Finding 8 — Constitutively active STAT6 mouse models recapitulate the human TH2/allergic phenotype

Two independent mouse models validate causality. The Stat6VT transgenic expresses a constitutively active STAT6 in T cells and "develop[s] spontaneous inflammation of the skin" (allergic dermatitis) plus allergic airway disease (PMID: 28653395). The patient-derived D419N knock-in mouse "elicited an abnormal TH2-dominant immune response in vivo, with findings similar to those observed in patients" (PMID: 40603028). Together, these models reproduce the cardinal human features (atopic skin disease, airway disease, TH2 skewing).

Evidence source: model organism (mouse).

Finding 9 — PARP14 links STAT6 GOF allergic disease to lymphomagenesis as a druggable co-activator

PARP14 (ARTD8) is an IL-4/STAT6-induced transcriptional co-activator: "the presence of interleukin-4 (IL-4) and activated Stat6 induces the enzymatic activity of PARP14 that promotes T helper type 2 differentiation and allergic airway disease" (PMID: 28653395). PARP14 is also "a novel target in STAT6 mutant follicular lymphoma" (PMID: 35851155). Because germline STAT6 GOF and somatic follicular-lymphoma STAT6 mutations affect the same DNA-binding-domain residues (notably D419), PARP14 represents a shared, druggable downstream node connecting the allergic and oncologic ends of the disease spectrum.

Evidence source: model organism + in vitro / cancer genomics.


Full Disease Characterization (15 Domains)

1. Disease Information

STAT6 GOF disease is a monogenic, autosomal-dominant primary atopic disorder / inborn error of immunity characterized by early-onset, severe, multi-system allergic disease driven by constitutive TH2 signaling. It was first defined as a distinct entity in 2023.

Identifier type Value
OMIM (disease) #620532 (Hyper-IgE syndrome 6, autosomal dominant, with recurrent infections; HIES6)
Mondo MONDO:0957807
GARD 0026874
MedGen 1851769
UMLS C5848786
NCIt C212086 (Activating STAT6 Gene Mutation)
Gene (OMIM) STAT6 601512
HGNC 11364
NCBI Gene 6778
UniProt P42226
Orphanet None dedicated identified
ICD-10/ICD-11 No specific code; mapped under primary immunodeficiency/atopic categories
MeSH No dedicated term; indexed via STAT6 / hyper-IgE / hypersensitivity

Synonyms/alternative names: STAT6 gain-of-function disease; STAT6-GOF; Hyper-IgE syndrome 6 (HIES6); autosomal dominant STAT6 GOF; STAT6-associated primary atopic disorder.

Information source type: Predominantly aggregated disease-level resources (OMIM, Mondo, HPO) built from a small number of individual-patient case cohorts/reports (n≈16 founding + additional single cases). This is a very rare, newly described disease, so all knowledge derives from individual patients described in the literature, not EHR-scale populations.

2. Etiology

  • Primary cause: germline heterozygous gain-of-function missense variants in STAT6. The disease is monogenic and genetic; no environmental or infectious cause is required.
  • Genetic risk factors: the causal variants themselves (DBD hotspot D419 and neighbors E372, E377, E382, D519). No modifier loci are established.
  • Environmental risk factors: none required for disease causation. Allergen exposure, as in common atopy, may trigger/exacerbate individual manifestations (food allergy, anaphylaxis, asthma), but the disease penetrates independent of specific exposures.
  • Protective factors: none established genetically or environmentally. Therapeutically, IL-4Rα blockade and JAK inhibition suppress the disease phenotype (see Section 12).
  • Gene–environment interactions: the hyperactive STAT6 axis lowers the threshold for TH2 responses to environmental allergens; thus environment shapes which allergic manifestations appear, while genotype drives the underlying diathesis. No formal GxE quantification exists.

3. Phenotypes

Quantitative HPO-annotated frequencies (n=16 founding cohort, PMID: 36884218):

Phenotype HPO term Frequency Type
Infantile onset HP:0003593 16/16 (100%) onset
Atopic dermatitis HP:0001047 15/16 (94%) clinical sign / skin
Food allergy HP:0500093 15/16 (94%) clinical sign
Increased eosinophil count HP:0001880 15/16 (94%) lab abnormality
Increased circulating IgE HP:0003212 present (high) lab abnormality
Asthma HP:0002099 11/16 (69%) clinical sign / respiratory
Gastrointestinal eosinophilia HP:0032064 10/16 (63%) lab / histopathology
Anaphylactic shock HP:0100845 9/16 (56%) clinical sign
Recurrent skin infections HP:0001581 7/16 (44%) clinical sign
Short stature HP:0004322 7/16 (44%) physical manifestation
Recurrent respiratory infections HP:0002205 5/16 (31%) clinical sign
Gastroesophageal reflux HP:0002020 4/16 (25%) clinical sign
Osteoporosis HP:0000939 3/16 (19%) lab / imaging
Recurrent viral infections HP:0004429 2/16 (13%) clinical sign
B-cell lymphoma HP:0012191 1/16 (6%) neoplasm
Eosinophilic esophagitis HP:0410151 present histopathology
Autosomal dominant inheritance HP:0000006 inheritance

Characteristics: age of onset is neonatal/infantile (100%); severity is generally severe (treatment-resistant atopic dermatitis); course is chronic/progressive with episodic anaphylaxis; variable expressivity is documented even within families (e.g., E377K kindred showed clinical heterogeneity, PMID: 36216080). Quality-of-life impact is substantial: severe pruritic dermatitis, dietary restriction from food allergy, anaphylaxis risk, and growth impairment—though formal EQ-5D/SF-36 data are not available for this rare disease.

4. Genetic/Molecular Information

  • Causal gene: STAT6 (12q13.3; OMIM 601512; HGNC:11364; NCBI Gene 6778; UniProt P42226).
  • Pathogenic variants (germline, dominant): E372K (c.1114G>A), E377K (c.1129G>A), E382Q (c.1144G>C), D419H (c.1255G>C), D419Y (c.1255G>T), D419G (c.1256A>G), D419N (c.1255G>A), D519H/N (c.1555G>C). Codon D419 is the recurrent hotspot.
  • Variant classification (ACMG/AMP, ClinVar): Pathogenic (E372K, E382Q, D419Y, D419G, D519H) or Likely pathogenic (D419H).
  • Variant type: exclusively missense to date.
  • Allele frequency: these variants are absent or ultra-rare in gnomAD; STAT6 is missense-constrained (mis_z = 3.47) and LoF-tolerant (pLI = 0.057, oe_lof upper = 0.54).
  • Somatic vs germline: the disease variants are germline; notably, somatic STAT6 DBD mutations at the same residues (D419) recur in follicular lymphoma.
  • Functional consequence: gain of function — constitutive and/or IL-4-hypersensitive STAT6 activation.
  • Modifier genes: none established. Epigenetic changes / chromosomal abnormalities: none reported; disease is a point-mutation disorder.

5. Environmental Information

No environmental toxin, occupational exposure, lifestyle factor, or infectious agent causes STAT6 GOF disease. Environmental allergens act as triggers for individual atopic manifestations. Recurrent infections (skin/respiratory/viral) reflect immune dysregulation intrinsic to the genotype rather than an environmental etiology.

6. Mechanism / Pathophysiology

Causal chain (upstream → downstream):

Germline STAT6 DBD missense variant (e.g., D419H/N, E372K)
│
▼
Constitutive / IL-4-hypersensitive STAT6 activation
  • sustained tyrosine phosphorylation (pSTAT6)
  • ligand-independent nuclear translocation (D419N, even unphosphorylated)
│
▼
Increased STAT6 target-gene transcription (e.g., PARP14, GATA3 program)
│
▼
Pathological TH2 skewing of CD4+ T cells (IL-4, IL-5, IL-13 ↑)
│
├──► B-cell IgE class switching  → hyper-IgE, food allergy, anaphylaxis
├──► Eosinophil recruitment/survival → hypereosinophilia, eosinophilic GI disease
├──► Skin barrier/Th2 inflammation → treatment-resistant atopic dermatitis
├──► Airway Th2 inflammation → asthma
└──► Chronic B-cell proliferation + PARP14 co-activation → follicular lymphoma risk
  • Molecular pathway: IL-4/IL-13 → JAK1/JAK2/TYK2 → STAT6 (KEGG JAK-STAT signaling; Reactome IL-4/IL-13 signaling). Upstream node = JAK kinases (JAK-inhibitor target); membrane receptor = IL-4Rα (dupilumab target).
  • Cellular processes: TH2 differentiation, IgE class-switch recombination, eosinophilia, type-2 inflammation.
  • Protein dysfunction: gain of function — enhanced DNA binding / nuclear retention of STAT6 (a transcription factor). Not misfolding or aggregation.
  • Immune involvement: immune dysregulation (allergy axis) with partial immunodeficiency (recurrent infections).
  • Transcriptional co-activator: PARP14 amplifies the STAT6/TH2 program and connects to lymphomagenesis.
  • Suggested GO terms: GO:0042092 (type 2 immune response), GO:0045064 (T-helper 2 cell differentiation), GO:0043330 (response to exogenous dsRNA — not applicable; use GO:0070670 response to IL-4), GO:0006357 (regulation of transcription by RNA Pol II), GO:0042113 (B-cell activation). Suggested CL terms: CL:0000546 (T-helper 2 cell), CL:0000236 (B cell), CL:0000771 (eosinophil), CL:0000097 (mast cell). Subcellular: GO:0005634 (nucleus) — the site of STAT6 dysfunction.

7. Anatomical Structures Affected

  • Primary organs / systems: skin (UBERON:0002097), immune/hematopoietic system (UBERON:0002405), gastrointestinal tract—esophagus (UBERON:0001043), stomach, gut—and respiratory system/lung (UBERON:0002048).
  • Secondary: skeletal system (short stature, osteoporosis); lymphoid tissue (lymphoma).
  • Tissues/cells: epithelial (skin/GI/airway barrier), and immune cell populations — TH2 cells (CL:0000546), eosinophils (CL:0000771), B cells/plasma cells (CL:0000236), mast cells.
  • Subcellular: nucleus (transcription-factor dysfunction).
  • Lateralization: systemic/bilateral (dermatitis, asthma); not lateralized.

8. Temporal Development

  • Onset: congenital/infantile (100%), insidious-to-chronic.
  • Progression: chronic, lifelong; atopic dermatitis is persistent and treatment-resistant; anaphylaxis is episodic; lymphoma is a late, rare complication.
  • Course: progressive multi-system atopy without treatment; treatment-induced remission/control achievable with dupilumab/JAK inhibitors.
  • Critical periods: early childhood — window for diagnosis and initiation of targeted therapy to prevent morbidity.

9. Inheritance and Population

  • Inheritance: autosomal dominant; ~70% sporadic/de novo (7/10 kindreds), ~30% inherited (3/10 kindreds) in the founding cohort.
  • Penetrance: appears high but with variable expressivity (intra-familial heterogeneity documented).
  • Epidemiology: ultra-rare; exact prevalence/incidence unknown (fewer than ~20 published families as of 2025). No founder effect, consanguinity role, or carrier-frequency data (dominant, de novo–enriched).
  • Demographics: reported across three continents; no ethnic predilection established; no clear sex ratio.

10. Diagnostics

  • Laboratory: markedly elevated serum total IgE (LOINC-mappable IgE assays), peripheral hypereosinophilia (CBC/differential), tissue eosinophilia on GI biopsy.
  • Biomarkers: STAT6 target-gene expression and pSTAT6 (functional readouts); TH2 cytokine skewing.
  • Genetic testing (definitive): whole-genome or whole-exome sequencing is the recommended upfront approach for primary atopic disorders ("Upfront genome-wide analysis by whole genome sequencing (WGS) will shorten the time to diagnosis", PMID: 39381601); targeted STAT6 single-gene or PAD gene-panel testing is an alternative. Functional confirmation (sustained pSTAT6, enhanced nuclear translocation, luciferase/EMSA reporter assays, patient PBMC signaling) distinguishes GOF variants from VUS.
  • Histopathology: eosinophilic infiltration of esophagus/GI tract; atopic dermatitis skin changes.
  • Differential diagnosis: other primary atopic disorders / transcription-factor IEIs — STAT3 loss-of-function (Job syndrome), FOXP3 deficiency (IPEX), T-bet deficiency, DOCK8 deficiency, Netherton syndrome (PMID: 37727514). STAT6 GOF is distinguished by the constitutive STAT6-activation signature and dupilumab responsiveness.
  • Screening: cascade genetic testing of at-risk relatives in inherited kindreds.

11. Outcome/Prognosis

  • Survival/mortality: no disease-specific mortality data; anaphylaxis and lymphoma are the principal life-threatening risks.
  • Morbidity: high — severe dermatitis, dietary restriction, growth impairment, recurrent infections; substantial quality-of-life burden (no formal EQ-5D/SF-36 data).
  • Complications: anaphylaxis, eosinophilic GI disease, recurrent infections, osteoporosis, and B-cell/follicular lymphoma (~6%).
  • Prognostic factors: the disease is highly treatment-responsive; early targeted therapy markedly improves outcomes. Lymphoma surveillance is warranted given the PARP14/STAT6 link.

12. Treatment

Therapy Class / target Mechanism Evidence MAXO
Dupilumab anti–IL-4Rα monoclonal antibody Blocks IL-4/IL-13 receptor upstream of STAT6 "highly effective improving both clinical manifestations and immunological biomarkers" (PMID: 36884218); effective for D519N (PMID: 40502541) MAXO monoclonal-antibody therapy
Ruxolitinib / JAK inhibitors JAK1/JAK2 inhibitor Reduces pSTAT6 by blocking upstream kinases "ruxolitinib reduced pSTAT6 levels in D419H HEK293T cells and patient PBMC" (PMID: 37316763) MAXO pharmacotherapy / targeted therapy
Supportive atopic care Topical steroids, emollients, allergen avoidance, epinephrine Symptom control Standard atopy management MAXO supportive care
PARP14 inhibition (experimental) small-molecule co-activator inhibitor Blocks downstream STAT6 co-activator; also anti-lymphoma Preclinical (PMID: 35851155; PMID: 28653395) MAXO experimental therapy

Personalized medicine: the disease is a paradigm of genotype-guided precision therapy — a druggable, hyperactive signaling axis directly matched to approved biologics (dupilumab) and JAK inhibitors. Pharmacogenomics: not specifically characterized. No gene/cell therapy is in clinical use.

13. Prevention

  • Primary prevention: none (monogenic, largely de novo). Genetic counseling for inherited kindreds; prenatal/preimplantation genetic testing is theoretically possible for known familial variants.
  • Secondary prevention: early genomic diagnosis and initiation of targeted therapy; allergen/anaphylaxis risk management.
  • Tertiary prevention: dupilumab/JAK inhibitors to prevent complications; lymphoma surveillance; infection prophylaxis as needed.
  • No immunization or population public-health intervention is applicable.

14. Other Species / Natural Disease

  • Taxonomy/orthologs: STAT6 is conserved; mouse Stat6 (NCBI Gene 20852). No naturally occurring companion-animal/wildlife equivalent of germline STAT6 GOF disease is catalogued (no OMIA entry identified). Comparative biology: the IL-4/STAT6/TH2 axis is evolutionarily conserved, underpinning the validity of mouse models. No zoonotic relevance.

15. Model Organisms

Model Type Genetic design Phenotype recapitulation Reference
Stat6VT Mouse (transgenic) Constitutively active STAT6 in T cells Spontaneous allergic skin inflammation + allergic airway disease; PARP14-dependent TH2 program PMID: 28653395
STAT6 D419N knock-in Mouse (patient-variant knock-in) Germline D419N "abnormal TH2-dominant immune response in vivo, with findings similar to those observed in patients" PMID: 40603028
Patient cells / HEK293T In vitro Overexpressed variant STAT6 pSTAT6 elevation, nuclear translocation, reporter activation; ruxolitinib response PMID: 37316763, PMID: 36884218
Gastric organoids In vitro (patient-derived) E377K Downstream effector-cytokine studies PMID: 36216080

Applications: mechanism of TH2 skewing, allergic skin/airway disease, target validation for dupilumab/JAK/PARP14. Limitations: mouse models capture allergic dermatitis and TH2 skewing but do not fully model the human lymphoma continuum or the complete multi-system phenotype.


Mechanistic Model / Interpretation

STAT6 GOF disease is best understood as a "single-node type-2 immune amplifier" disorder. A germline missense change in the STAT6 DNA-binding domain converts a normally ligand-controlled transcription factor into a hyperactive or constitutively active driver of the TH2 gene program. The location of the mutations is mechanistically decisive: the DBD hotspot (D419) either stabilizes STAT6 in a DNA-bound/nuclear-retained state or lowers the activation threshold for IL-4 signaling. This produces the entire downstream cascade of type-2 immunity—IgE class switching, eosinophilia, and barrier-tissue inflammation—explaining why one gene defect yields such a broad, coherent, multi-organ atopic phenotype.

Three lines of evidence converge on gain-of-function rather than haploinsufficiency: (1) the dominant inheritance with recurrent, clustered missense variants; (2) gnomAD constraint showing LoF tolerance but strong missense intolerance (mis_z = 3.47); and (3) direct functional assays showing sustained/ligand-independent STAT6 activation. The mouse models close the causal loop: constitutively active STAT6 alone is sufficient to produce spontaneous allergic skin and airway disease.

The disease also illuminates a shared germline–somatic axis. The identical DBD residues mutated germline in this atopic disorder are recurrently mutated somatically in follicular lymphoma, and PARP14 functions as a common downstream co-activator in both settings. This explains the small but real lymphoma risk and nominates PARP14 as a mechanistic bridge and therapeutic target spanning allergy and oncology.

Clinically, the model is directly actionable: blocking the axis at the receptor (dupilumab/IL-4Rα) or upstream kinase (JAK inhibitor) reverses both symptoms and biomarkers, making STAT6 GOF disease a textbook example of precision medicine in inborn errors of immunity.


Evidence Base

PMID Title (abbrev.) Contribution
36884218 Human germline heterozygous GOF STAT6 variants cause severe allergic disease Defining cohort (n=16): GOF mechanism, AD inheritance, core phenotype, dupilumab efficacy
36216080 A germline STAT6 GOF variant is associated with early-onset allergies E377K DBD variant; spontaneous STAT6 activation; gastric organoids; variable expressivity
36758835 Severe allergic dysregulation due to a GOF mutation in STAT6 E372K DBD variant
37316763 Autosomal dominant STAT6 GOF causes severe atopy associated with lymphoma D419H variant; ruxolitinib reduces pSTAT6; follicular lymphoma link
40603028 Mechanism of pathogenesis by a GOF STAT6 variant D419N: ligand-independent nuclear translocation; knock-in mouse recapitulation
40502541 STAT6 GOF: p.D519N responds to dupilumab New variant; expands phenotype; dupilumab response
38238227 Human germline GOF STAT6: from allergy to lymphoma Review; allergy-to-lymphoma spectrum; targeted-treatment overview
37727514 Transcription factor defects in IEIs with atopy Places STAT6 GOF among TF-defect atopic IEIs; differential diagnosis
39381601 Rapid identification of PAD by upfront genomic sequencing Diagnostic strategy: upfront WGS for primary atopic disorders
28653395 PARP14 limits severity of allergic skin disease Stat6VT mouse; PARP14 as STAT6 co-activator in TH2/allergic disease
35851155 PARP14 is a novel target in STAT6 mutant follicular lymphoma PARP14 druggability; germline–somatic mechanistic bridge

All eleven papers are mutually consistent; none challenge the core GOF model. Evidence spans human clinical/genetic cohorts, in vitro functional assays, and two mouse models, providing multi-modal validation.


Limitations and Knowledge Gaps

  1. Very small sample size. Fewer than ~20 families are published; frequencies (e.g., lymphoma 6%) derive from n=16 and carry wide confidence intervals. True prevalence/incidence is unknown.
  2. No dedicated Orphanet/ICD code, complicating registry-based epidemiology.
  3. Penetrance and expressivity are incompletely quantified; intra-familial heterogeneity is described but not modeled.
  4. Long-term outcomes (life expectancy, lymphoma lifetime risk, treatment durability) are unknown given the disease's recency.
  5. Genotype–phenotype correlations (e.g., whether specific DBD residues predict lymphoma vs pure atopy) are not yet resolved.
  6. No formal QoL instruments, pharmacogenomics, or gene/cell-therapy data.
  7. PARP14 inhibition remains preclinical for this indication.

Proposed Follow-up Experiments / Actions

  1. Establish an international STAT6-GOF registry to refine prevalence, penetrance, lymphoma risk, and natural history.
  2. Systematic genotype–phenotype mapping across all reported variants (D419 hotspot vs others) to test whether specific residues predict lymphoma risk or dupilumab responsiveness.
  3. Prospective dupilumab and JAK-inhibitor trials with standardized clinical and biomarker (pSTAT6, IgE, eosinophil) endpoints and QoL instruments (EQ-5D, PROMIS).
  4. Lymphoma surveillance protocol development, leveraging the shared germline–somatic DBD/PARP14 axis.
  5. PARP14 inhibitor preclinical testing in the D419N knock-in mouse for both allergic and lymphoma endpoints.
  6. Deep functional characterization of each variant (constitutive vs ligand-hypersensitive) to guide therapy selection (receptor blockade vs kinase inhibition).
  7. Assign a dedicated Orphanet/ICD-11 code and complete HPO annotation for downstream variants.

Artifacts