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1
Inheritance
5
Pathophys.
11
Phenotypes
2
Gaps
10
Pathograph
1
Genes
6
Medical Actions
3
Differentials
1
References
1
Deep Research
🏷

Classifications

Harrison's Chapter
IMMUNE_RHEUMATOLOGIC ONCOLOGY_HEMATOLOGY
👪

Inheritance

1
Somatic mosaicism (not inherited) HP:0001442
VEXAS is caused by acquired somatic (post-zygotic, mosaic) UBA1 variants and is not a heritable Mendelian disease. There is no germline transmission to offspring and no recurrence risk in families. The strong male predominance reflects the X-linked location of UBA1 (single-X dosage in males); affected females typically require acquired monosomy X, skewed X-inactivation, or a second somatic event.
Typified by somatic mosaicism
Show evidence (1 reference)
PMID:40373178 SUPPORT Human Clinical
"To date, all identified pathogenic variants are acquired (i.e., postzygotic) and lineage restricted in the blood. No confirmed occurrences of vertical transmission or sib recurrence have been reported."
GeneReviews confirms the somatic, non-heritable nature of VEXAS with no vertical transmission or sibling recurrence.
?

Discussions and Knowledge Gaps

2
Do existing zebrafish and mouse Uba1-perturbation models faithfully reproduce the full multi-organ, relapsing human VEXAS syndrome (chondritis, neutrophilic skin disease, vacuolated marrow precursors, and clonal evolution to MDS), or only its molecular/inflammatory arm?
HUMAN MODEL MISMATCH OPEN vexas_model_human_fidelity
Animal and cellular models reproduce the proximal ubiquitylation defect, UPR/innate-immune activation, and myeloid bias well, but no single model reproduces the age-dependent somatic-clonal acquisition or the human-specific UBA1b cytoplasmic-isoform start-codon architecture at Met41 that underlies the human multi-organ syndrome. Translational fidelity to the human clinical phenotype therefore remains open.
Proposed experiments
Humanized hematopoietic-restricted somatic Met41 mouse model
vexas_humanized_met41_mouse
Engineer humanized, hematopoietic-restricted somatic Met41 mouse models with age-dependent clonal acquisition and assess multi-organ phenotype recapitulation including marrow precursor vacuolization and MDS evolution.
What are the general-population incidence and finalized formal diagnostic criteria for VEXAS syndrome?
KNOWLEDGE GAP OPEN vexas_population_incidence_criteria
Attached to
disease#VEXAS Syndrome
Prevalence is estimated from a single US regional, predominantly White health-system cohort; general-population incidence and validated consensus diagnostic criteria are not yet established, and diverse-ancestry data are sparse.

Pathophysiology

5
Somatic UBA1 Met41 Mutation in Hematopoietic Stem Cells
The founding lesion of VEXAS is an acquired (post-zygotic, mosaic) somatic mutation in UBA1 affecting methionine-41 (p.Met41), arising in hematopoietic stem and progenitor cells during adult life. Because UBA1 is X-linked, a single somatic hit in males is sufficient to reach a pathogenic mutant allele fraction. The mutation is detectable in peripheral-blood myeloid cells but not in lymphocytes or fibroblasts.
Hematopoietic stem cell CL:0000037
Show evidence (2 references)
PMID:33108101 SUPPORT Human Clinical
"We identified 25 men with somatic mutations affecting methionine-41 (p.Met41) in UBA1, the major E1 enzyme that initiates ubiquitylation."
Establishes the defining somatic UBA1 p.Met41 lesion in affected men as the founding genetic event.
PMID:33108101 SUPPORT Human Clinical
"Mutations were found in more than half the hematopoietic stem cells, including peripheral-blood myeloid cells but not lymphocytes or fibroblasts."
Localizes the somatic mutation to hematopoietic stem cells and the myeloid compartment, supporting the HSC origin and diagnostic tissue restriction.
Loss of Cytoplasmic UBA1 and Reduced Ubiquitylation
Mutations at p.Met41 abolish initiation of the canonical cytoplasmic UBA1 isoform (UBA1b) and force expression of a novel, catalytically impaired isoform initiated at a downstream methionine (p.Met67). The net effect is a global reduction in cytoplasmic ubiquitylation, the obligatory first step of the ubiquitin-proteasome system. The level of residual UBA1b translation is genotype-dependent and tracks with disease severity and survival.
Protein ubiquitination GO:0016567 ↓ DECREASED
Show evidence (2 references)
PMID:33108101 SUPPORT Human Clinical
"Mutations affecting p.Met41 resulted in loss of the canonical cytoplasmic isoform of UBA1 and in expression of a novel, catalytically impaired isoform initiated at p.Met67."
Documents the isoform switch from cytoplasmic UBA1b to a catalytically impaired p.Met67-initiated isoform as the proximal molecular consequence.
PMID:35793467 SUPPORT In Vitro
"Using in vitro models and patient-derived cells, we demonstrate that p.Met41Val variant supports less UBA1b translation than either p.Met41Leu or p.Met41Thr, providing a molecular rationale for decreased survival."
Shows that residual cytoplasmic UBA1b translation is genotype-dependent and mechanistically linked to prognosis.
Innate Immune Activation
In UBA1-mutant peripheral-blood and myeloid cells, decreased ubiquitylation activates cellular stress responses, including the unfolded protein response, and engages multiple innate immune pathways (NF-kB, type I interferon, and inflammasome signaling), producing the cytokine-driven autoinflammatory state. VEXAS is a prototypic innate-driven (autoinflammatory) disease rather than a classic adaptive autoimmune disease.
Monocyte CL:0000576
Inflammatory response GO:0006954 ↑ INCREASED
Show evidence (2 references)
PMID:33108101 SUPPORT In Vitro
"Mutant peripheral-blood cells showed decreased ubiquitylation and activated innate immune pathways."
Directly links reduced ubiquitylation in mutant cells to activation of innate immune pathways underlying the autoinflammatory phenotype.
PMID:33108101 SUPPORT Model Organism
"Knockout of the cytoplasmic UBA1 isoform homologue in zebrafish caused systemic inflammation."
Zebrafish knockout of the cytoplasmic UBA1 homologue recapitulates systemic inflammation, supporting the causal mechanism in vivo.
Multi-Organ Neutrophilic Inflammation
The cytokine-driven inflammatory program produces recurrent, multi-organ neutrophilic inflammation: neutrophilic and leukocytoclastic cutaneous lesions, auricular and nasal chondritis, neutrophilic pulmonary inflammation, scleritis/uveitis, and vasculitis. This effector phase is the clinical face of the autoinflammatory arm.
Neutrophil CL:0000775
Show evidence (1 reference)
PMID:33108101 SUPPORT Human Clinical
"an often fatal, treatment-refractory inflammatory syndrome develops in late adulthood, with fevers, cytopenias, characteristic vacuoles in myeloid and erythroid precursor cells, dysplastic bone marrow, neutrophilic cutaneous and pulmonary inflammation, chondritis, and vasculitis."
Enumerates the multi-organ neutrophilic inflammatory manifestations driven by the disease.
Myeloid-Biased Dysplastic Hematopoiesis
The UBA1-mutant clone, originating in hematopoietic stem cells, expands with a myeloid bias and produces dysplastic hematopoiesis. The pathognomonic morphologic readout is cytoplasmic vacuolization of myeloid and erythroid precursor cells in the bone marrow; the hematologic trajectory frequently progresses to myelodysplastic syndrome and is accompanied by macrocytic anemia and cytopenias.
Erythroid lineage cell CL:0000764
Show evidence (1 reference)
PMID:33108101 SUPPORT Human Clinical
"characteristic vacuoles in myeloid and erythroid precursor cells, dysplastic bone marrow"
Documents the precursor vacuolization and dysplastic marrow that define the hematologic arm of VEXAS.

Pathograph

Use the checkboxes to hide or show graph categories. Hover nodes for evidence and cross-linked metadata.
Pathograph: causal mechanism network for VEXAS Syndrome Interactive directed graph showing how pathophysiology mechanisms, phenotypes, genetic factors and variants, experimental models, environmental triggers, and treatments relate through causal and linked edges.

Phenotypes

11
Blood 4
Macrocytic Anemia VERY_FREQUENT Macrocytic anemia HP:0001972
Course: PROGRESSIVE
Show evidence (1 reference)
PMID:36692560 SUPPORT Human Clinical
"all individuals had anemia (hemoglobin: mean, 7.8 g/dL; median, 7.5 g/dL), which was mostly macrocytic (10/11"
Genome-first cohort shows anemia in all carriers, macrocytic in 10/11 (91%), supporting macrocytic anemia as a near-universal (VERY_FREQUENT) feature.
Thrombocytopenia VERY_FREQUENT Thrombocytopenia HP:0001873
Show evidence (1 reference)
PMID:36692560 SUPPORT Human Clinical
"with concomitant thrombocytopenia (10/11"
Genome-first cohort documents concomitant thrombocytopenia in 10/11 (91%) of carriers.
Myelodysplastic Syndrome Myelodysplasia HP:0002863
Show evidence (1 reference)
PMID:33108101 SUPPORT Human Clinical
"Most of these 25 patients met clinical criteria for an inflammatory syndrome (relapsing polychondritis, Sweet's syndrome, polyarteritis nodosa, or giant-cell arteritis) or a hematologic condition (myelodysplastic syndrome or multiple myeloma) or both."
Documents myelodysplastic syndrome (and multiple myeloma) as hematologic conditions met by patients with VEXAS.
Venous Thromboembolism Deep venous thrombosis HP:0002625
Show evidence (1 reference)
PMID:40373178 SUPPORT Human Clinical
"recurrent chondritis, arthritis, pan ocular inflammation, and unprovoked venous thrombosis."
GeneReviews lists unprovoked venous thrombosis among the most common inflammatory findings.
Eye 1
Scleritis Scleritis HP:0100532
Show evidence (1 reference)
PMID:40373178 SUPPORT Human Clinical
"The most common inflammatory findings include recurrent fever, skin lesions, pulmonary infiltrates, recurrent chondritis, arthritis, pan ocular inflammation, and unprovoked venous thrombosis."
GeneReviews lists pan ocular inflammation among the most common inflammatory findings; scleritis is a characteristic ocular manifestation.
Metabolism 1
Recurrent Fever Recurrent fever HP:0001954
Temporal: RECURRENT
Show evidence (1 reference)
PMID:33108101 SUPPORT Human Clinical
"an often fatal, treatment-refractory inflammatory syndrome develops in late adulthood, with fevers, cytopenias"
Lists fevers among the cardinal features of the late-onset inflammatory syndrome.
Musculoskeletal 1
Arthritis Arthritis HP:0001369
Show evidence (1 reference)
PMID:40373178 SUPPORT Human Clinical
"recurrent fever, skin lesions, pulmonary infiltrates, recurrent chondritis, arthritis, pan ocular inflammation"
GeneReviews lists arthritis among the common inflammatory findings.
Respiratory 1
Pulmonary Infiltrates Pulmonary infiltrates HP:0002113
Show evidence (1 reference)
PMID:33108101 SUPPORT Human Clinical
"neutrophilic cutaneous and pulmonary inflammation, chondritis, and vasculitis."
Documents neutrophilic pulmonary inflammation as a manifestation.
Other 3
Neutrophilic Dermatosis VERY_FREQUENT Neutrophilic infiltration of the skin HP:0031234
Show evidence (2 references)
PMID:38865133 SUPPORT Human Clinical
"skin involvement was common (93"
Cohort of 112 patients shows skin involvement in 93/112 (83%) and as the most frequent presenting feature, supporting VERY_FREQUENT. Note the band reflects overall skin involvement; neutrophilic dermatosis was the predominant histopathologic pattern (next evidence item).
PMID:38865133 SUPPORT Human Clinical
"predominant skin histopathologic findings were leukocytoclastic vasculitis"
Documents leukocytoclastic vasculitis and neutrophilic dermatosis as predominant skin histopathology.
Cutaneous Leukocytoclastic Vasculitis Leukocytoclastic vasculitis HP:0034786
Show evidence (1 reference)
PMID:38865133 SUPPORT Human Clinical
"the p.Met41Val variant was associated with vasculitic lesions"
Documents vasculitic skin lesions associated with the p.Met41Val genotype.
Chondritis Chondritis HP:0100662
Temporal: RECURRENT
Show evidence (1 reference)
PMID:33108101 SUPPORT Human Clinical
"neutrophilic cutaneous and pulmonary inflammation, chondritis, and vasculitis."
Lists chondritis among the characteristic inflammatory manifestations.
🧬

Genetic Associations

1
UBA1 (Somatic (post-zygotic, mosaic) mutations in UBA1 (Xp11.23), predominantly at p.Met41 (p.Met41Thr, p.Met41Val, p.Met41Leu) and at splice/non-Met41 sites that also impair cytoplasmic UBA1b, are the defining cause of VEXAS. The variants are restricted to the hematopoietic compartment and absent in skin fibroblasts. Genotype influences phenotype and prognosis: p.Met41Val carries the worst survival and least residual UBA1b, whereas p.Met41Leu carries the best. )
Gene: UBA1 hgnc:12469 relationship_type: CAUSATIVE variant_origin: SOMATIC
Show evidence (2 references)
PMID:35793467 SUPPORT Human Clinical
"We analyzed 83 patients with somatic pathogenic variants in UBA1 at p.Met41 (p.Met41Leu/Thr/Val), the start codon for translation of the cytoplasmic isoform of UBA1 (UBA1b)."
Defines the three canonical p.Met41 somatic genotypes at the cytoplasmic UBA1b start codon.
PMID:35793467 SUPPORT Human Clinical
"ear chondritis was associated with increased survival, whereas transfusion dependence and the p.Met41Val variant were independently associated with decreased survival."
Establishes p.Met41Val as an independent predictor of decreased survival, supporting genotype-phenotype-prognosis correlation.
💊

Medical Actions

6
Glucocorticoid Therapy
Action: Pharmacotherapy NCIT:C15986
Agent: prednisone CHEBI:8382
Glucocorticoids (e.g., prednisone) are first-line and almost universally effective for inflammatory manifestations, but VEXAS is typically steroid-dependent and chronic high-dose exposure drives the need for steroid-sparing agents.
Show evidence (1 reference)
PMID:38865133 SUPPORT Human Clinical
"Oral prednisone improved skin manifestations in 67 of 73 patients"
Documents high response of skin manifestations to oral prednisone.
Ruxolitinib (JAK Inhibitor)
Action: Pharmacotherapy NCIT:C15986
Agent: ruxolitinib CHEBI:66919
Among JAK inhibitors, the JAK1/2 inhibitor ruxolitinib is the most effective in VEXAS, with clinical remissions and steroid reduction in the majority of treated patients.
Mechanism Target:
INHIBITS Innate Immune Activation — JAK1/2 inhibition suppresses the innate immune / cytokine signaling that drives the autoinflammatory phenotype.
Show evidence (1 reference)
PMID:35609174 SUPPORT Human Clinical
"encouraging evidence supporting the use of the JAK1/2 inhibitor ruxolitinib with clinical remissions and reductions in steroid use seen in the majority of patients."
Retrospective multicenter study supports ruxolitinib efficacy with remissions and steroid reduction in most patients.
Tocilizumab (IL-6 Inhibition)
Action: Pharmacotherapy NCIT:C15986
Agent: Tocilizumab NCIT:C84217
The anti-IL-6 receptor monoclonal antibody tocilizumab is used as a steroid-sparing agent with partial efficacy.
Mechanism Target:
INHIBITS Innate Immune Activation — IL-6 receptor blockade dampens the cytokine-driven inflammatory program.
Show evidence (1 reference)
PMID:40373178 SUPPORT Human Clinical
"second-line steroid-sparing agents including interleukin (IL)-6 inhibitors, Janus kinase inhibitors (JAKi), and anti-IL-1 therapies."
GeneReviews lists IL-6 inhibitors among second-line steroid-sparing agents.
Azacitidine (Hypomethylating Agent)
Action: chemotherapy MAXO:0000647
Agent: azacitidine CHEBI:2038
The hypomethylating agent azacitidine targets the UBA1-mutant hematopoietic population, used particularly in patients with concurrent MDS, and can occasionally induce molecular remission of the UBA1 clone.
Mechanism Target:
INHIBITS Myeloid-Biased Dysplastic Hematopoiesis — Hypomethylating therapy targets the dysplastic, UBA1-mutant myeloid population.
Show evidence (1 reference)
PMID:40373178 SUPPORT Human Clinical
"hypomethylating agents like azacitidine are used to treat individuals with VEXAS syndrome with concurrent MDS with varying success."
GeneReviews documents azacitidine use for VEXAS with concurrent MDS.
Allogeneic Hematopoietic Stem Cell Transplantation
Action: allogeneic hematopoietic stem cell transplantation MAXO:0001479
Allogeneic HSCT is currently the only potentially curative therapy; it eradicates the UBA1-mutant clone but carries considerable transplant-related morbidity and mortality and is reserved for selected patients.
Mechanism Target:
INHIBITS Somatic UBA1 Met41 Mutation in Hematopoietic Stem Cells — Replacement of the patient's hematopoietic system eradicates the UBA1-mutant clone, the founding lesion.
Show evidence (1 reference)
PMID:40373178 SUPPORT Human Clinical
"Allogeneic hematopoietic stem cell transplantation (HSCT) is currently the only curative treatment for VEXAS syndrome"
GeneReviews identifies allogeneic HSCT as the only curative therapy.
Anakinra (IL-1 Inhibition)
Action: Pharmacotherapy NCIT:C15986
Agent: anakinra CHEBI:231683
Anakinra, a recombinant IL-1 receptor antagonist, is used as an anti-IL-1 steroid-sparing option but has limited efficacy in VEXAS. Importantly, it frequently causes severe injection-site reactions in VEXAS patients, a disease-specific safety signal.
Mechanism Target:
INHIBITS Innate Immune Activation — IL-1 receptor antagonism dampens IL-1-driven autoinflammatory signaling.
Show evidence (2 references)
PMID:40373178 SUPPORT Human Clinical
"second-line steroid-sparing agents including interleukin (IL)-6 inhibitors, Janus kinase inhibitors (JAKi), and anti-IL-1 therapies."
GeneReviews lists anti-IL-1 therapies among second-line steroid-sparing agents.
PMID:38865133 SUPPORT Human Clinical
"Patients with VEXAS treated with anakinra frequently developed severe injection-site reactions"
Documents the disease-specific anakinra injection-site reaction safety signal in VEXAS patients.
🔬

Biochemical Markers

1
Elevated C-reactive protein (Positive)
🔀

Differential Diagnoses

3

Conditions with similar clinical presentations that must be differentiated from VEXAS Syndrome:

Overlapping Features A substantial fraction of older men diagnosed with relapsing polychondritis in fact have VEXAS; the somatic UBA1 mutation, marrow vacuoles, and macrocytic anemia distinguish VEXAS.
Overlapping Features VEXAS skin lesions frequently resemble (histiocytoid) Sweet syndrome; accompanying macrocytic anemia and UBA1 testing distinguish VEXAS.
Myelodysplastic syndrome without autoinflammation
Overlapping Features MDS in an older man with prominent systemic inflammation should prompt UBA1 testing for VEXAS.
{ }

Source YAML

click to show
name: VEXAS Syndrome
creation_date: "2026-06-29T00:00:00Z"
category: Complex
disease_term:
  preferred_term: VEXAS syndrome
  term:
    id: MONDO:0026777
    label: VEXAS syndrome
parents:
  - autoinflammatory syndrome
  - rare disease
classifications:
  harrisons_chapter:
  - classification_value: IMMUNE_RHEUMATOLOGIC
  - classification_value: ONCOLOGY_HEMATOLOGY
description: >
  VEXAS (Vacuoles, E1 enzyme, X-linked, Autoinflammatory, Somatic) syndrome is a
  severe, late-onset, treatment-refractory systemic autoinflammatory and
  hematologic disease caused by acquired somatic mutations in UBA1, the X-linked
  gene encoding the major E1 ubiquitin-activating enzyme. The mutations arise in
  hematopoietic stem and progenitor cells and predominantly affect
  methionine-41 (p.Met41), the start codon for the catalytically active
  cytoplasmic UBA1 isoform (UBA1b); their loss forces translation of a
  catalytically impaired isoform from a downstream start site, crippling
  cytoplasmic ubiquitylation. Because UBA1 is X-linked, the disease
  overwhelmingly affects men (about 96% of patients), with onset typically after
  age 50. It bridges rheumatology and hematology, combining systemic
  inflammation (recurrent fever, neutrophilic dermatosis, chondritis,
  vasculitis, pulmonary infiltrates, ocular inflammation, venous thrombosis)
  with myeloid-biased hematologic abnormalities (macrocytic anemia,
  characteristic cytoplasmic vacuoles in myeloid and erythroid precursors,
  thrombocytopenia, and frequent progression to myelodysplastic syndrome). VEXAS
  unified several previously idiopathic adult inflammatory presentations
  (relapsing polychondritis, Sweet syndrome, polyarteritis nodosa, giant-cell
  arteritis) under a single somatic molecular cause.
synonyms:
  - VEXAS
  - vacuoles, E1 enzyme, X-linked, autoinflammatory, somatic syndrome
  - UBA1-related autoinflammatory disease
references:
  - reference: PMID:40373178
    title: "VEXAS Syndrome."
    tags:
      - GeneReviews
pathophysiology:
- name: Somatic UBA1 Met41 Mutation in Hematopoietic Stem Cells
  description: >
    The founding lesion of VEXAS is an acquired (post-zygotic, mosaic) somatic
    mutation in UBA1 affecting methionine-41 (p.Met41), arising in hematopoietic
    stem and progenitor cells during adult life. Because UBA1 is X-linked, a
    single somatic hit in males is sufficient to reach a pathogenic mutant
    allele fraction. The mutation is detectable in peripheral-blood myeloid
    cells but not in lymphocytes or fibroblasts.
  cell_types:
  - preferred_term: Hematopoietic stem cell
    term:
      id: CL:0000037
      label: hematopoietic stem cell
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "We identified 25 men with somatic mutations affecting methionine-41 (p.Met41) in UBA1, the major E1 enzyme that initiates ubiquitylation."
    explanation: >
      Establishes the defining somatic UBA1 p.Met41 lesion in affected men as
      the founding genetic event.
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "Mutations were found in more than half the hematopoietic stem cells, including peripheral-blood myeloid cells but not lymphocytes or fibroblasts."
    explanation: >
      Localizes the somatic mutation to hematopoietic stem cells and the myeloid
      compartment, supporting the HSC origin and diagnostic tissue restriction.
  downstream:
  - target: Loss of Cytoplasmic UBA1 and Reduced Ubiquitylation
    causal_link_type: DIRECT
    description: >
      Loss of the p.Met41 start codon abolishes translation of the cytoplasmic
      UBA1b isoform, driving expression of a catalytically impaired isoform and
      reduced ubiquitylation.
- name: Loss of Cytoplasmic UBA1 and Reduced Ubiquitylation
  description: >
    Mutations at p.Met41 abolish initiation of the canonical cytoplasmic UBA1
    isoform (UBA1b) and force expression of a novel, catalytically impaired
    isoform initiated at a downstream methionine (p.Met67). The net effect is a
    global reduction in cytoplasmic ubiquitylation, the obligatory first step of
    the ubiquitin-proteasome system. The level of residual UBA1b translation is
    genotype-dependent and tracks with disease severity and survival.
  biological_processes:
  - preferred_term: Protein ubiquitination
    term:
      id: GO:0016567
      label: protein ubiquitination
    modifier: DECREASED
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "Mutations affecting p.Met41 resulted in loss of the canonical cytoplasmic isoform of UBA1 and in expression of a novel, catalytically impaired isoform initiated at p.Met67."
    explanation: >
      Documents the isoform switch from cytoplasmic UBA1b to a catalytically
      impaired p.Met67-initiated isoform as the proximal molecular consequence.
  - reference: PMID:35793467
    reference_title: "Translation of cytoplasmic UBA1 contributes to VEXAS syndrome pathogenesis."
    supports: SUPPORT
    evidence_source: IN_VITRO
    snippet: "Using in vitro models and patient-derived cells, we demonstrate that p.Met41Val variant supports less UBA1b translation than either p.Met41Leu or p.Met41Thr, providing a molecular rationale for decreased survival."
    explanation: >
      Shows that residual cytoplasmic UBA1b translation is genotype-dependent
      and mechanistically linked to prognosis.
  downstream:
  - target: Innate Immune Activation
    causal_link_type: DIRECT
    description: >
      Reduced cytoplasmic ubiquitylation triggers cellular stress responses and
      activates innate immune signaling in mutant myeloid cells.
- name: Innate Immune Activation
  description: >
    In UBA1-mutant peripheral-blood and myeloid cells, decreased ubiquitylation
    activates cellular stress responses, including the unfolded protein response,
    and engages multiple innate immune pathways (NF-kB, type I interferon, and
    inflammasome signaling), producing the cytokine-driven autoinflammatory
    state. VEXAS is a prototypic innate-driven (autoinflammatory) disease rather
    than a classic adaptive autoimmune disease.
  cell_types:
  - preferred_term: Monocyte
    term:
      id: CL:0000576
      label: monocyte
  biological_processes:
  - preferred_term: Inflammatory response
    term:
      id: GO:0006954
      label: inflammatory response
    modifier: INCREASED
  notes: >
    The cited NEJM abstract supports activation of innate immune pathways as an
    umbrella. The more specific downstream signals reported in the full text and
    later mechanistic work — unfolded protein response (UPR), canonical NF-kB
    signaling, type I interferon signature, and inflammasome activation — are
    described in the node prose but are not asserted as evidenced GO modifiers
    here because the cached abstract does not itemize them; add them with
    citable snippets if those specific signals are quoted from a fetched source.
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: IN_VITRO
    snippet: "Mutant peripheral-blood cells showed decreased ubiquitylation and activated innate immune pathways."
    explanation: >
      Directly links reduced ubiquitylation in mutant cells to activation of
      innate immune pathways underlying the autoinflammatory phenotype.
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: MODEL_ORGANISM
    snippet: "Knockout of the cytoplasmic UBA1 isoform homologue in zebrafish caused systemic inflammation."
    explanation: >
      Zebrafish knockout of the cytoplasmic UBA1 homologue recapitulates
      systemic inflammation, supporting the causal mechanism in vivo.
  downstream:
  - target: Multi-Organ Neutrophilic Inflammation
    causal_link_type: DIRECT
    description: >
      Innate immune activation drives recurrent neutrophilic inflammation across
      skin, cartilage, lung, eye, and vasculature.
  - target: Myeloid-Biased Dysplastic Hematopoiesis
    causal_link_type: DIRECT
    description: >
      The UBA1-mutant clone drives myeloid-biased, dysplastic hematopoiesis with
      characteristic precursor vacuolization and progression to MDS.
- name: Multi-Organ Neutrophilic Inflammation
  description: >
    The cytokine-driven inflammatory program produces recurrent, multi-organ
    neutrophilic inflammation: neutrophilic and leukocytoclastic cutaneous
    lesions, auricular and nasal chondritis, neutrophilic pulmonary
    inflammation, scleritis/uveitis, and vasculitis. This effector phase is the
    clinical face of the autoinflammatory arm.
  cell_types:
  - preferred_term: Neutrophil
    term:
      id: CL:0000775
      label: neutrophil
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "an often fatal, treatment-refractory inflammatory syndrome develops in late adulthood, with fevers, cytopenias, characteristic vacuoles in myeloid and erythroid precursor cells, dysplastic bone marrow, neutrophilic cutaneous and pulmonary inflammation, chondritis, and vasculitis."
    explanation: >
      Enumerates the multi-organ neutrophilic inflammatory manifestations
      driven by the disease.
- name: Myeloid-Biased Dysplastic Hematopoiesis
  description: >
    The UBA1-mutant clone, originating in hematopoietic stem cells, expands with
    a myeloid bias and produces dysplastic hematopoiesis. The pathognomonic
    morphologic readout is cytoplasmic vacuolization of myeloid and erythroid
    precursor cells in the bone marrow; the hematologic trajectory frequently
    progresses to myelodysplastic syndrome and is accompanied by macrocytic
    anemia and cytopenias.
  cell_types:
  - preferred_term: Erythroid lineage cell
    term:
      id: CL:0000764
      label: erythroid lineage cell
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "characteristic vacuoles in myeloid and erythroid precursor cells, dysplastic bone marrow"
    explanation: >
      Documents the precursor vacuolization and dysplastic marrow that define
      the hematologic arm of VEXAS.
phenotypes:
- category: Hematologic
  name: Macrocytic Anemia
  description: >
    Macrocytic anemia is a near-universal hematologic feature of VEXAS and is
    often progressive and transfusion-dependent.
  phenotype_term:
    preferred_term: Macrocytic anemia
    term:
      id: HP:0001972
      label: Macrocytic anemia
    clinical_course: PROGRESSIVE
  frequency: VERY_FREQUENT
  evidence:
  - reference: PMID:36692560
    reference_title: "Estimated Prevalence and Clinical Manifestations of UBA1 Variants Associated With VEXAS Syndrome in a Clinical Population."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "all individuals had anemia (hemoglobin: mean, 7.8 g/dL; median, 7.5 g/dL), which was mostly macrocytic (10/11"
    explanation: >
      Genome-first cohort shows anemia in all carriers, macrocytic in 10/11
      (91%), supporting macrocytic anemia as a near-universal (VERY_FREQUENT)
      feature.
- category: Hematologic
  name: Thrombocytopenia
  description: >
    Thrombocytopenia frequently accompanies the macrocytic anemia and dysplastic
    hematopoiesis.
  frequency: VERY_FREQUENT
  phenotype_term:
    preferred_term: Thrombocytopenia
    term:
      id: HP:0001873
      label: Thrombocytopenia
  evidence:
  - reference: PMID:36692560
    reference_title: "Estimated Prevalence and Clinical Manifestations of UBA1 Variants Associated With VEXAS Syndrome in a Clinical Population."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "with concomitant thrombocytopenia (10/11"
    explanation: >
      Genome-first cohort documents concomitant thrombocytopenia in 10/11 (91%)
      of carriers.
- category: Hematologic
  name: Myelodysplastic Syndrome
  description: >
    A substantial fraction of patients develop myelodysplastic syndrome, mostly
    lower-risk, reflecting clonal evolution of the UBA1-mutant population.
  phenotype_term:
    preferred_term: Myelodysplasia
    term:
      id: HP:0002863
      label: Myelodysplasia
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "Most of these 25 patients met clinical criteria for an inflammatory syndrome (relapsing polychondritis, Sweet's syndrome, polyarteritis nodosa, or giant-cell arteritis) or a hematologic condition (myelodysplastic syndrome or multiple myeloma) or both."
    explanation: >
      Documents myelodysplastic syndrome (and multiple myeloma) as hematologic
      conditions met by patients with VEXAS.
- category: Constitutional
  name: Recurrent Fever
  description: >
    Recurrent fevers are a cardinal manifestation of the systemic
    autoinflammatory phenotype.
  phenotype_term:
    preferred_term: Recurrent fever
    term:
      id: HP:0001954
      label: Recurrent fever
    temporality: RECURRENT
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "an often fatal, treatment-refractory inflammatory syndrome develops in late adulthood, with fevers, cytopenias"
    explanation: >
      Lists fevers among the cardinal features of the late-onset inflammatory
      syndrome.
- category: Dermatologic
  name: Neutrophilic Dermatosis
  description: >
    Skin involvement is common and is frequently the presenting feature, with
    neutrophilic dermal infiltrates (often resembling histiocytoid Sweet
    syndrome), leukocytoclastic vasculitis, and perivascular dermatitis.
  phenotype_term:
    preferred_term: Neutrophilic dermatosis
    term:
      id: HP:0031234
      label: Neutrophilic infiltration of the skin
  frequency: VERY_FREQUENT
  evidence:
  - reference: PMID:38865133
    reference_title: "Skin Manifestations of VEXAS Syndrome and Associated Genotypes."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "skin involvement was common (93"
    explanation: >
      Cohort of 112 patients shows skin involvement in 93/112 (83%) and as the
      most frequent presenting feature, supporting VERY_FREQUENT. Note the band
      reflects overall skin involvement; neutrophilic dermatosis was the
      predominant histopathologic pattern (next evidence item).
  - reference: PMID:38865133
    reference_title: "Skin Manifestations of VEXAS Syndrome and Associated Genotypes."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "predominant skin histopathologic findings were leukocytoclastic vasculitis"
    explanation: >
      Documents leukocytoclastic vasculitis and neutrophilic dermatosis as
      predominant skin histopathology.
- category: Dermatologic
  name: Cutaneous Leukocytoclastic Vasculitis
  description: >
    Leukocytoclastic vasculitis is a frequent cutaneous histopathologic pattern,
    particularly associated with the p.Met41Val genotype.
  phenotype_term:
    preferred_term: Leukocytoclastic vasculitis
    term:
      id: HP:0034786
      label: Leukocytoclastic vasculitis
  evidence:
  - reference: PMID:38865133
    reference_title: "Skin Manifestations of VEXAS Syndrome and Associated Genotypes."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "the p.Met41Val variant was associated with vasculitic lesions"
    explanation: >
      Documents vasculitic skin lesions associated with the p.Met41Val
      genotype.
- category: Musculoskeletal
  name: Chondritis
  description: >
    Relapsing auricular and nasal chondritis is a common manifestation; a large
    fraction of older men diagnosed with relapsing polychondritis in fact have
    VEXAS.
  phenotype_term:
    preferred_term: Chondritis
    term:
      id: HP:0100662
      label: Chondritis
    temporality: RECURRENT
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "neutrophilic cutaneous and pulmonary inflammation, chondritis, and vasculitis."
    explanation: >
      Lists chondritis among the characteristic inflammatory manifestations.
- category: Respiratory
  name: Pulmonary Infiltrates
  description: >
    Neutrophilic pulmonary inflammation with pulmonary infiltrates (and
    organizing pneumonia, pleural effusions) is a frequent organ manifestation.
  phenotype_term:
    preferred_term: Pulmonary infiltrates
    term:
      id: HP:0002113
      label: Pulmonary infiltrates
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "neutrophilic cutaneous and pulmonary inflammation, chondritis, and vasculitis."
    explanation: >
      Documents neutrophilic pulmonary inflammation as a manifestation.
- category: Ophthalmologic
  name: Scleritis
  description: >
    Ocular inflammation, including scleritis, episcleritis, uveitis, and
    periorbital/orbital inflammation, occurs in a substantial minority of
    patients.
  phenotype_term:
    preferred_term: Scleritis
    term:
      id: HP:0100532
      label: Scleritis
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "The most common inflammatory findings include recurrent fever, skin lesions, pulmonary infiltrates, recurrent chondritis, arthritis, pan ocular inflammation, and unprovoked venous thrombosis."
    explanation: >
      GeneReviews lists pan ocular inflammation among the most common
      inflammatory findings; scleritis is a characteristic ocular manifestation.
- category: Vascular
  name: Venous Thromboembolism
  description: >
    Unprovoked venous thromboembolism (deep venous thrombosis and pulmonary
    embolism) is a frequent and clinically important complication.
  phenotype_term:
    preferred_term: Deep venous thrombosis
    term:
      id: HP:0002625
      label: Deep venous thrombosis
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "recurrent chondritis, arthritis, pan ocular inflammation, and unprovoked venous thrombosis."
    explanation: >
      GeneReviews lists unprovoked venous thrombosis among the most common
      inflammatory findings.
- category: Musculoskeletal
  name: Arthritis
  description: >
    Inflammatory arthritis and polyarthralgia are common musculoskeletal
    manifestations.
  phenotype_term:
    preferred_term: Arthritis
    term:
      id: HP:0001369
      label: Arthritis
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "recurrent fever, skin lesions, pulmonary infiltrates, recurrent chondritis, arthritis, pan ocular inflammation"
    explanation: >
      GeneReviews lists arthritis among the common inflammatory findings.
biochemical:
- name: Elevated C-reactive protein
  biomarker_term:
    preferred_term: Elevated circulating C-reactive protein concentration
    term:
      id: HP:0011227
      label: Elevated circulating C-reactive protein concentration
  presence: Positive
  notes: >
    Persistently elevated acute-phase reactants (C-reactive protein, erythrocyte
    sedimentation rate) reflect the chronic systemic inflammatory state.
    Near-universal in active VEXAS but non-specific; the defining laboratory clue
    is macrocytic anemia with elevated acute-phase reactants in an older man.
genetic:
- name: UBA1
  gene_term:
    preferred_term: UBA1
    term:
      id: hgnc:12469
      label: UBA1
  variant_origin: SOMATIC
  relationship_type: CAUSATIVE
  association: >
    Somatic (post-zygotic, mosaic) mutations in UBA1 (Xp11.23), predominantly at
    p.Met41 (p.Met41Thr, p.Met41Val, p.Met41Leu) and at splice/non-Met41 sites
    that also impair cytoplasmic UBA1b, are the defining cause of VEXAS. The
    variants are restricted to the hematopoietic compartment and absent in skin
    fibroblasts. Genotype influences phenotype and prognosis: p.Met41Val carries
    the worst survival and least residual UBA1b, whereas p.Met41Leu carries the
    best.
  evidence:
  - reference: PMID:35793467
    reference_title: "Translation of cytoplasmic UBA1 contributes to VEXAS syndrome pathogenesis."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "We analyzed 83 patients with somatic pathogenic variants in UBA1 at p.Met41 (p.Met41Leu/Thr/Val), the start codon for translation of the cytoplasmic isoform of UBA1 (UBA1b)."
    explanation: >
      Defines the three canonical p.Met41 somatic genotypes at the cytoplasmic
      UBA1b start codon.
  - reference: PMID:35793467
    reference_title: "Translation of cytoplasmic UBA1 contributes to VEXAS syndrome pathogenesis."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "ear chondritis was associated with increased survival, whereas transfusion dependence and the p.Met41Val variant were independently associated with decreased survival."
    explanation: >
      Establishes p.Met41Val as an independent predictor of decreased survival,
      supporting genotype-phenotype-prognosis correlation.
inheritance:
- name: Somatic mosaicism (not inherited)
  inheritance_term:
    preferred_term: Typified by somatic mosaicism
    term:
      id: HP:0001442
      label: Typified by somatic mosaicism
  description: >
    VEXAS is caused by acquired somatic (post-zygotic, mosaic) UBA1 variants and
    is not a heritable Mendelian disease. There is no germline transmission to
    offspring and no recurrence risk in families. The strong male predominance
    reflects the X-linked location of UBA1 (single-X dosage in males); affected
    females typically require acquired monosomy X, skewed X-inactivation, or a
    second somatic event.
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "To date, all identified pathogenic variants are acquired (i.e., postzygotic) and lineage restricted in the blood. No confirmed occurrences of vertical transmission or sib recurrence have been reported."
    explanation: >
      GeneReviews confirms the somatic, non-heritable nature of VEXAS with no
      vertical transmission or sibling recurrence.
prevalence:
- population: Men older than 50 years (US regional health system, genome-first ascertainment)
  measure_type: POINT_PREVALENCE
  prevalence_class: BAND_1_5_PER_10000
  rate_per_100000: 23.42469
  percentage: 1 in 4269
  evidence:
  - reference: PMID:36692560
    reference_title: "Estimated Prevalence and Clinical Manifestations of UBA1 Variants Associated With VEXAS Syndrome in a Clinical Population."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "1 in 4269 men older than 50 years"
    explanation: >
      Genome-first Geisinger MyCode study estimates disease-associated UBA1
      variant prevalence at 1 in 4269 men older than 50 years.
- population: Women older than 50 years (US regional health system, genome-first ascertainment)
  measure_type: POINT_PREVALENCE
  prevalence_class: BAND_1_9_PER_100000
  rate_per_100000: 3.811266
  percentage: 1 in 26238
  evidence:
  - reference: PMID:36692560
    reference_title: "Estimated Prevalence and Clinical Manifestations of UBA1 Variants Associated With VEXAS Syndrome in a Clinical Population."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "1 in 26 238 women older than 50 years"
    explanation: >
      Same study estimates a much lower prevalence in women older than 50 years,
      consistent with the X-linked male predominance.
diagnosis:
- name: Molecular genetic testing for somatic UBA1 variants
  description: >
    Diagnosis is established by identifying a somatic UBA1 pathogenic variant by
    molecular genetic testing of peripheral blood and/or bone marrow aspirate
    (myeloid-enriched fractions increase sensitivity), but not skin fibroblasts.
    Because the variant allele fraction is often high, exome sequencing can
    misread the somatic variant as hemizygous germline; confirming absence in
    non-hematopoietic tissue establishes the somatic (mosaic) state.
  diagnosis_term:
    preferred_term: molecular genetic testing
    term:
      id: MAXO:0000533
      label: molecular genetic testing
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "a UBA1 somatic (also known as mosaic or postzygotic) pathogenic variant identified by molecular genetic testing in peripheral blood and/or bone marrow aspirate, but not skin fibroblasts."
    explanation: >
      GeneReviews specifies the confirmatory molecular test and the diagnostic
      tissue restriction (blood/marrow, not fibroblasts).
  - reference: PMID:36038944
    reference_title: "Exome sequencing can misread high variant allele fraction of somatic variants in UBA1 as hemizygous in VEXAS syndrome: a case report."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "Sequencing of different tissues should be considered when there is conflict between the UBA1 variant status and the clinical findings."
    explanation: >
      Highlights the exome misinterpretation pitfall and the need to sequence
      multiple tissues to confirm somatic status.
- name: Bone marrow examination for precursor vacuolization
  description: >
    Bone marrow aspirate classically shows cytoplasmic vacuoles in myeloid and
    erythroid precursor cells, a highly suggestive morphologic clue, alongside
    myeloid hyperplasia and dysplasia.
  diagnosis_term:
    preferred_term: bone marrow examination
    term:
      id: MAXO:0000753
      label: bone marrow examination
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "vacuoles in myeloid and erythroid precursor cells."
    explanation: >
      GeneReviews lists the characteristic precursor vacuolization seen on bone
      marrow examination.
differential_diagnoses:
- name: Relapsing polychondritis
  description: >
    A substantial fraction of older men diagnosed with relapsing polychondritis
    in fact have VEXAS; the somatic UBA1 mutation, marrow vacuoles, and
    macrocytic anemia distinguish VEXAS.
- name: Sweet syndrome
  description: >
    VEXAS skin lesions frequently resemble (histiocytoid) Sweet syndrome;
    accompanying macrocytic anemia and UBA1 testing distinguish VEXAS.
- name: Myelodysplastic syndrome without autoinflammation
  description: >
    MDS in an older man with prominent systemic inflammation should prompt UBA1
    testing for VEXAS.
treatments:
- name: Glucocorticoid Therapy
  description: >
    Glucocorticoids (e.g., prednisone) are first-line and almost universally
    effective for inflammatory manifestations, but VEXAS is typically
    steroid-dependent and chronic high-dose exposure drives the need for
    steroid-sparing agents.
  therapeutic_modality: SMALL_MOLECULE
  treatment_term:
    preferred_term: Pharmacotherapy
    term:
      id: NCIT:C15986
      label: Pharmacotherapy
    therapeutic_agent:
    - preferred_term: prednisone
      term:
        id: CHEBI:8382
        label: prednisone
  evidence:
  - reference: PMID:38865133
    reference_title: "Skin Manifestations of VEXAS Syndrome and Associated Genotypes."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "Oral prednisone improved skin manifestations in 67 of 73 patients"
    explanation: >
      Documents high response of skin manifestations to oral prednisone.
- name: Ruxolitinib (JAK Inhibitor)
  description: >
    Among JAK inhibitors, the JAK1/2 inhibitor ruxolitinib is the most effective
    in VEXAS, with clinical remissions and steroid reduction in the majority of
    treated patients.
  therapeutic_modality: SMALL_MOLECULE
  treatment_term:
    preferred_term: Pharmacotherapy
    term:
      id: NCIT:C15986
      label: Pharmacotherapy
    therapeutic_agent:
    - preferred_term: ruxolitinib
      term:
        id: CHEBI:66919
        label: ruxolitinib
  target_mechanisms:
  - target: Innate Immune Activation
    treatment_effect: INHIBITS
    description: >
      JAK1/2 inhibition suppresses the innate immune / cytokine signaling that
      drives the autoinflammatory phenotype.
  evidence:
  - reference: PMID:35609174
    reference_title: "Ruxolitinib is more effective than other JAK inhibitors to treat VEXAS syndrome: a retrospective multicenter study."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "encouraging evidence supporting the use of the JAK1/2 inhibitor ruxolitinib with clinical remissions and reductions in steroid use seen in the majority of patients."
    explanation: >
      Retrospective multicenter study supports ruxolitinib efficacy with
      remissions and steroid reduction in most patients.
- name: Tocilizumab (IL-6 Inhibition)
  description: >
    The anti-IL-6 receptor monoclonal antibody tocilizumab is used as a
    steroid-sparing agent with partial efficacy.
  therapeutic_modality: MONOCLONAL_ANTIBODY
  treatment_term:
    preferred_term: Pharmacotherapy
    term:
      id: NCIT:C15986
      label: Pharmacotherapy
    therapeutic_agent:
    - preferred_term: Tocilizumab
      term:
        id: NCIT:C84217
        label: Tocilizumab
  target_mechanisms:
  - target: Innate Immune Activation
    treatment_effect: INHIBITS
    description: >
      IL-6 receptor blockade dampens the cytokine-driven inflammatory program.
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "second-line steroid-sparing agents including interleukin (IL)-6 inhibitors, Janus kinase inhibitors (JAKi), and anti-IL-1 therapies."
    explanation: >
      GeneReviews lists IL-6 inhibitors among second-line steroid-sparing
      agents.
- name: Azacitidine (Hypomethylating Agent)
  description: >
    The hypomethylating agent azacitidine targets the UBA1-mutant hematopoietic
    population, used particularly in patients with concurrent MDS, and can
    occasionally induce molecular remission of the UBA1 clone.
  therapeutic_modality: SMALL_MOLECULE
  treatment_term:
    preferred_term: chemotherapy
    term:
      id: MAXO:0000647
      label: chemotherapy
    therapeutic_agent:
    - preferred_term: azacitidine
      term:
        id: CHEBI:2038
        label: 5-azacytidine
  target_mechanisms:
  - target: Myeloid-Biased Dysplastic Hematopoiesis
    treatment_effect: INHIBITS
    description: >
      Hypomethylating therapy targets the dysplastic, UBA1-mutant myeloid
      population.
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "hypomethylating agents like azacitidine are used to treat individuals with VEXAS syndrome with concurrent MDS with varying success."
    explanation: >
      GeneReviews documents azacitidine use for VEXAS with concurrent MDS.
- name: Allogeneic Hematopoietic Stem Cell Transplantation
  description: >
    Allogeneic HSCT is currently the only potentially curative therapy; it
    eradicates the UBA1-mutant clone but carries considerable transplant-related
    morbidity and mortality and is reserved for selected patients.
  therapeutic_modality: CELL_THERAPY
  treatment_term:
    preferred_term: allogeneic hematopoietic stem cell transplantation
    term:
      id: MAXO:0001479
      label: allogeneic hematopoietic stem cell transplantation
  target_mechanisms:
  - target: Somatic UBA1 Met41 Mutation in Hematopoietic Stem Cells
    treatment_effect: INHIBITS
    description: >
      Replacement of the patient's hematopoietic system eradicates the
      UBA1-mutant clone, the founding lesion.
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "Allogeneic hematopoietic stem cell transplantation (HSCT) is currently the only curative treatment for VEXAS syndrome"
    explanation: >
      GeneReviews identifies allogeneic HSCT as the only curative therapy.
- name: Anakinra (IL-1 Inhibition)
  description: >
    Anakinra, a recombinant IL-1 receptor antagonist, is used as an anti-IL-1
    steroid-sparing option but has limited efficacy in VEXAS. Importantly, it
    frequently causes severe injection-site reactions in VEXAS patients, a
    disease-specific safety signal.
  therapeutic_modality: PROTEIN_REPLACEMENT
  treatment_term:
    preferred_term: Pharmacotherapy
    term:
      id: NCIT:C15986
      label: Pharmacotherapy
    therapeutic_agent:
    - preferred_term: anakinra
      term:
        id: CHEBI:231683
        label: Anakinra
  target_mechanisms:
  - target: Innate Immune Activation
    treatment_effect: INHIBITS
    description: >
      IL-1 receptor antagonism dampens IL-1-driven autoinflammatory signaling.
  evidence:
  - reference: PMID:40373178
    reference_title: "VEXAS Syndrome."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "second-line steroid-sparing agents including interleukin (IL)-6 inhibitors, Janus kinase inhibitors (JAKi), and anti-IL-1 therapies."
    explanation: >
      GeneReviews lists anti-IL-1 therapies among second-line steroid-sparing
      agents.
  - reference: PMID:38865133
    reference_title: "Skin Manifestations of VEXAS Syndrome and Associated Genotypes."
    supports: SUPPORT
    evidence_source: HUMAN_CLINICAL
    snippet: "Patients with VEXAS treated with anakinra frequently developed severe injection-site reactions"
    explanation: >
      Documents the disease-specific anakinra injection-site reaction safety
      signal in VEXAS patients.
animal_models:
- species: Danio rerio (zebrafish)
  genotype: Cytoplasmic UBA1 isoform homologue knockout (CRISPR-Cas9)
  description: >
    CRISPR-Cas9 knockout of the cytoplasmic UBA1 isoform homologue in zebrafish
    causes systemic inflammation, providing in vivo support for the proximal
    ubiquitylation-loss mechanism driving autoinflammation.
  evidence:
  - reference: PMID:33108101
    reference_title: "Somatic Mutations in UBA1 and Severe Adult-Onset Autoinflammatory Disease."
    supports: SUPPORT
    evidence_source: MODEL_ORGANISM
    snippet: "Knockout of the cytoplasmic UBA1 isoform homologue in zebrafish caused systemic inflammation."
    explanation: >
      Zebrafish model recapitulates systemic inflammation downstream of
      cytoplasmic UBA1 loss.
discussions:
- discussion_id: vexas_model_human_fidelity
  kind: HUMAN_MODEL_MISMATCH
  status: OPEN
  attaches_to:
  - pathophysiology#Multi-Organ Neutrophilic Inflammation
  prompt: >
    Do existing zebrafish and mouse Uba1-perturbation models faithfully
    reproduce the full multi-organ, relapsing human VEXAS syndrome (chondritis,
    neutrophilic skin disease, vacuolated marrow precursors, and clonal
    evolution to MDS), or only its molecular/inflammatory arm?
  rationale: >
    Animal and cellular models reproduce the proximal ubiquitylation defect,
    UPR/innate-immune activation, and myeloid bias well, but no single model
    reproduces the age-dependent somatic-clonal acquisition or the human-specific
    UBA1b cytoplasmic-isoform start-codon architecture at Met41 that underlies
    the human multi-organ syndrome. Translational fidelity to the human clinical
    phenotype therefore remains open.
  proposed_experiments:
  - experiment_id: vexas_humanized_met41_mouse
    name: Humanized hematopoietic-restricted somatic Met41 mouse model
    description: >
      Engineer humanized, hematopoietic-restricted somatic Met41 mouse models
      with age-dependent clonal acquisition and assess multi-organ phenotype
      recapitulation including marrow precursor vacuolization and MDS evolution.
- discussion_id: vexas_population_incidence_criteria
  kind: KNOWLEDGE_GAP
  status: OPEN
  attaches_to:
  - disease#VEXAS Syndrome
  prompt: >
    What are the general-population incidence and finalized formal diagnostic
    criteria for VEXAS syndrome?
  rationale: >
    Prevalence is estimated from a single US regional, predominantly White
    health-system cohort; general-population incidence and validated consensus
    diagnostic criteria are not yet established, and diverse-ancestry data are
    sparse.
notes: >
  VEXAS is a clonal-hematopoietic autoinflammatory disorder bridging
  rheumatology and hematology, defined by somatic UBA1 p.Met41 mutations. No
  existing dismech mechanism module maps cleanly to its somatic-clonal /
  type-I-interferon-adjacent innate-immune-dysregulation pattern, so no
  conforms_to edge is asserted; a future clonal-hematopoiesis or
  interferonopathy module would be the natural conformance target. The repo's
  Relapsing_Polychondritis entry already models the VEXAS overlap from the RP
  side. Some clinical details (precise organ-specific frequencies, plasma-cell
  dyscrasia, aseptic meningitis, orchitis) are documented in the literature but
  were not added as separate phenotype nodes where a verified exact-substring
  snippet for the specific claim was not available.
📚

References & Deep Research

References

1
VEXAS Syndrome.
No top-level findings curated for this source.

Deep Research

1
Claude Code
1. Disease Information
claude-haiku-4-5-20251001, claude-opus-4-8[1m] 10 citations 2026-06-29T11:09:58.072764

1. Disease Information

Overview. VEXAS syndrome is a severe, adult-onset, treatment-refractory autoinflammatory disease driven by acquired (somatic) loss-of-function mutations in the X-linked gene UBA1, the apex enzyme of the ubiquitylation cascade. The mutation arises in hematopoietic stem and progenitor cells (HSPCs), so it sits at the crossroads of autoinflammation and clonal hematologic disease (myelodysplastic syndrome, plasma-cell dyscrasias). The name is an acronym coined in the discovery paper:

Vacuoles, E1 enzyme, X-linked, Autoinflammatory, Somatic — Beck DB et al., NEJM 2020 (PMID:33108101).

It is best understood as a clonal hematopoietic disorder masquerading as, and overlapping with, a host of rheumatologic syndromes (relapsing polychondritis, Sweet syndrome, polyarteritis nodosa, giant cell arteritis, undifferentiated systemic inflammation). It unified many previously "idiopathic" adult inflammatory presentations under a single molecular cause.

Key identifiers. - MONDO: MONDO:0026777 - OMIM: #301054 (VEXAS SYNDROME) - Orphanet: ORPHA:596753 - GARD: 15001 - MeSH: indexed under "VEXAS syndrome" (introduced ~2022) - ICD-10/ICD-11: No dedicated code yet; typically coded under autoinflammatory/myelodysplastic categories (ICD-10 D89.9 / D46.x). ICD-11 has no specific stem code as of this writing — (data gap).

Synonyms / alternative names. "UBA1-related autoinflammatory disease"; "Somatic UBA1-mutation–associated autoinflammatory syndrome"; historically subsumed under "relapsing polychondritis with myelodysplasia," "Sweet syndrome with MDS," and "idiopathic adult-onset autoinflammatory disease."

Data derivation. Knowledge is a mix: deep-phenotyped disease-level cohorts (NIH/NHGRI, French GFEV, multicenter registries) plus a landmark genome-first / EHR-linked population study (Geisinger MyCode, PMID:36692560) that ascertained patients from sequencing rather than clinic — an unusual and valuable "reverse" ascertainment for a rare disease.

Sources: NEJM 2020 (PMID:33108101) · GeneReviews NBK614471 · OMIM 301054


2. Etiology

Primary cause (genetic, somatic). VEXAS is caused by somatic (post-zygotic, mosaic) mutations in UBA1 acquired in hematopoietic stem cells during adult life — it is not inherited and not a germline disease. The canonical mutations hit codon 41 (p.Met41), which is the alternative translation-initiation start codon for the cytoplasmic UBA1b isoform. Loss of Met41 abolishes cytoplasmic UBA1b initiation; cells instead make a catalytically impaired, mislocalized isoform (UBA1c) from a downstream start site, crippling cytoplasmic ubiquitylation.

"We identified 25 men who had somatic mutations in UBA1... The mutations were found in peripheral-blood cells... the somatic mutations affected methionine-41 (p.Met41)." — Beck DB et al., NEJM 2020 (PMID:33108101). (HUMAN_CLINICAL)

Risk factors. - Age: Strongest determinant. Disease is essentially adult-only, median onset mid-60s; risk rises with age (consistent with age-related clonal hematopoiesis as the soil for acquiring the UBA1 mutation). - Sex (male): Because UBA1 is X-linked, males (one X) need only a single somatic hit to reach a pathogenic mutant allele fraction. Males ≈96% of cases. - Clonal hematopoiesis: VEXAS is mechanistically a form of clonal hematopoiesis; co-occurring DNMT3A and TET2 mutations are common and may precede or accompany the UBA1 clone. - Genetic risk in females: Females generally require an additional event — acquired monosomy X (loss of the wild-type X), X-inactivation skewing, or a second somatic hit — to manifest, which explains their rarity. (PMID:33108101; GeneReviews NBK614471).

Protective factors. No established environmental protective factors. The closest "protective" genetic concept is the mutation-type gradient: p.Met41Leu (which preserves more residual UBA1b translation) carries markedly better survival than p.Met41Val. Higher residual wild-type/UBA1b activity is protective at the cellular level (PMID:35793465, Ferrada/Beck Blood 2022, IN_VITRO + HUMAN_CLINICAL).

Gene–environment interactions. No proven exogenous trigger. The dominant "environment" is endogenous aging hematopoiesis providing the clonal substrate. Infection/inflammation can precipitate flares but is not a documented cause. (Largely a data gap for true GxE.)


3. Phenotypes

VEXAS is multisystem. Frequencies below are pooled from GeneReviews and major cohorts (NEJM 2020, JAMA 2023, French cohort). Mark these as HUMAN_CLINICAL.

Constitutional / inflammatory - Recurrent fevers — 65–90%. HPO: HP:0001954 (Recurrent fever) / HP:0011947. Episodic, often weekly; adult onset; recurrent. - Weight loss / cachexia, fatigue, malaise — very frequent. HP:0001824 (Weight loss).

Skin (≈80%, often the presenting feature) - Neutrophilic dermatosis / Sweet-syndrome–like lesions — dominant pattern. HPO: HP:0200035 (Neutrophilic dermatosis) / HP:0000962 (Hyperkeratosis – not apt); best: HP:0200035. - Cutaneous vasculitis, leukocytoclastic vasculitis — HP:0011008 / HP:0025476 (Cutaneous small vessel vasculitis). - Skin biopsy classically shows a leukocytoclastic and neutrophilic/histiocytoid infiltrate with myeloid precursors carrying the UBA1 mutation.

Cartilage / musculoskeletal - Relapsing chondritis (auricular and nasal) — 36–54%. HPO: HP:0002770 (Chondritis) / HP:0100786 (auricular). A large fraction of "relapsing polychondritis" in older men is actually VEXAS. - Inflammatory arthritis / polyarthralgia — 28–58%. HP:0001369 (Arthritis).

Eye (30–46%) - Periorbital edema, scleritis, episcleritis, uveitis, orbital inflammation — HPO: HP:0100534 (Scleritis), HP:0000554 (Uveitis), HP:0100539 (Periorbital edema).

Lung (35–55%) - Pulmonary infiltrates, organizing pneumonia, pleural effusions, neutrophilic alveolitis — HPO: HP:0006530 (Abnormal pulmonary interstitial morphology) / HP:0002113 (Pulmonary infiltrates) / HP:0002202 (Pleural effusion).

Vascular / thrombotic (23–41%) - Venous thromboembolism (DVT/PE) predominant; some arterial. HPO: HP:0002625 (Deep venous thrombosis), HP:0002204 (Pulmonary embolism), HP:0001907 (Thromboembolism). Episodic/recurrent.

Hematologic (near-universal) - Macrocytic anemia — ~97%. HPO: HP:0001972 (Macrocytic anemia) / HP:0001903 (Anemia). Progressive, transfusion-dependent in many. - Cytoplasmic vacuoles in myeloid and erythroid precursors (bone marrow) — the pathognomonic morphologic clue. HPO: closest is HP:0011273 (Abnormal myeloid cell morphology) — (no precise "vacuolated precursor" HP term; data gap). - Thrombocytopenia — 10–48%. HP:0001873. - Myelodysplastic syndrome (MDS) — 31–53% (mostly low/very-low risk). HP:0002863 (Myelodysplasia). - Plasma-cell dyscrasia (MGUS / multiple myeloma) — 10–25%. HP:0012184 (Abnormal circulating immunoglobulin) / monoclonal gammopathy. - Markedly elevated CRP/ESR — near-universal. HP:0011227 (Elevated C-reactive protein level), HP:0003565 (Elevated erythrocyte sedimentation rate).

Other - Orchitis/epididymitis, aseptic meningitis, gastrointestinal inflammation, hearing loss reported less commonly.

Onset / severity / progression / QoL. Onset adult (median ~66 y). Course is chronic, relapsing-remitting with progressive cumulative organ damage; severity moderate-to-severe and frequently glucocorticoid-dependent. QoL impact is high: chronic high-dose steroid exposure, transfusion dependence, recurrent hospitalization, and substantial fatigue/pain burden. Formal EQ-5D/SF-36 data are sparse — (QoL instrument data gap).


4. Genetic / Molecular Information

Causal gene. UBA1 (ubiquitin-like modifier-activating enzyme 1; E1 enzyme). HGNC: HGNC:12469 (dismech CURIE form hgnc:12469); NCBI Gene 7317; Xp11.23; OMIM gene 314370. Encodes the sole or principal E1 that charges ubiquitin with ATP and hands it to E2 conjugating enzymes — the obligatory first step of essentially all cellular ubiquitylation.

Pathogenic variants (somatic, X-linked). - Canonical codon-41 variants (≈80–90% of cases): - p.Met41Thr — c.122T>C — most common; associated with more ocular inflammation; ~83% 5-yr survival. - p.Met41Val — c.121A>G — most aggressive; less chondritis, more undifferentiated systemic inflammation, worst survival (~60–77% 5-yr); lowest residual UBA1b. - p.Met41Leu — c.121A>C — frequent skin/Sweet phenotype; best survival (~100% 5-yr). - Splice and non-Met41 variants: e.g., c.118-1G>C, c.118-2A>C (splice-site), p.Ser56Phe, p.Gly477Ala, and others that also impair cytoplasmic UBA1b — these broaden the variant spectrum and are recognized in later cohorts (Poulter JA et al., Blood 2021, PMID:33690795; and subsequent series). (HUMAN_CLINICAL / IN_VITRO)

Classification. Pathogenic / likely pathogenic per functional + segregation-with-disease evidence; these are somatic mosaic calls, so ACMG germline rules apply imperfectly — interpretation hinges on variant allele fraction (VAF) and functional data.

Variant origin & allele fraction. Somatic, not germline. Restricted to the hematopoietic compartment (blood/marrow), absent in skin fibroblasts — a key diagnostic discriminator. VAF ranges ~4–95%, typically high in peripheral myeloid cells; the mutation enriches in myeloid lineage over time.

Population frequency. Not present in germline population databases (gnomAD) as a constitutional variant — it is an acquired somatic event, so "allele frequency" is age- and tissue-dependent rather than a fixed population number.

Functional consequence. Loss of cytoplasmic UBA1b → global reduction in cytoplasmic ubiquitylation (a partial loss-of-function with downstream gain-of-inflammatory-function at the cellular level). Met41 is the AUG start for the catalytically active cytoplasmic isoform; its loss forces use of a downstream Met67 start producing the dysfunctional UBA1c.

"Translation of cytoplasmic UBA1 contributes to VEXAS syndrome pathogenesis... patients with p.Met41Val have... lower residual translation of the normal cytoplasmic UBA1 isoform UBA1b." — Ferrada/Beck et al., Blood 2022 (PMID:35793465). (IN_VITRO + HUMAN_CLINICAL)

Modifier genes. Co-occurring clonal mutations — DNMT3A, TET2 (clonal hematopoiesis), and MDS-associated genes — modify hematologic trajectory and malignant risk.

Epigenetics. No primary epigenetic cause; however, the therapeutic efficacy of hypomethylating agents (azacitidine) implies DNA-methylation–sensitive clonal biology. Direct methylome studies are limited — (data gap).

Chromosomal abnormalities. Acquired monosomy X / loss of wild-type X is an important mechanism enabling disease in females and can accompany clonal evolution in males.


5. Environmental Information

  • Environmental/toxic factors: None established as causal. (Data gap.)
  • Lifestyle factors: No proven dietary/smoking/alcohol contribution to onset; smoking and cardiovascular risk factors are relevant only to thrombotic-complication management.
  • Infectious agents: No infectious cause. Infections are a leading cause of death in VEXAS (immunosuppression + cytopenias), and intercurrent infection can trigger flares — but VEXAS is not an infectious disease. NCBI Taxonomy: not applicable.

The "environmental" driver is essentially endogenous somatic mutagenesis in aging hematopoiesis.


6. Mechanism / Pathophysiology

Causal chain (upstream → downstream):

  1. Somatic UBA1 p.Met41 mutation in an HSPC → loss of cytoplasmic UBA1b → global reduction in cytoplasmic ubiquitylation. (initiating lesion; IN_VITRO + HUMAN_CLINICAL, PMID:33108101, PMID:35793465)
  2. Impaired ubiquitin–proteasome protein quality controlER stress and activation of the unfolded protein response (UPR) and dysregulated autophagy in mutant myeloid cells.
  3. Innate immune activation: mutant monocytes/myeloid cells show inflammasome activation, NF-κB and type I/II interferon signatures, and elevated IL-6, IL-1β, TNF-α. Defective Lys63/Met1 (linear) polyubiquitylation of inflammatory signaling complexes dysregulates death/inflammation checkpoints.

"Mutant cells showed decreased ubiquitylation [activating] cellular stress responses that lead to upregulation of the unfolded-protein response... and a shared gene expression signature consistent with the activation of multiple innate immune pathways." — Beck DB et al., NEJM 2020 (PMID:33108101). (IN_VITRO)

  1. Myeloid bias and dysplastic hematopoiesis: UBA1-mutant clones outcompete in the myeloid lineage; recent work shows inflammation and myeloid bias can arise via partly independent mechanisms downstream of UBA1 loss (Nature 2025, s41586-025-09815-0). The cytoplasmic vacuoles in marrow precursors are a morphologic readout of this proteostatic/autophagic stress.
  2. Aberrant regulated cell death: Uba1-mutant macrophages undergo RIPK1/RIPK3-linked inflammatory cell death, amplifying sterile inflammation (biorxiv 2025; mechanistic literature). (MODEL_ORGANISM / IN_VITRO)
  3. Clinical output: chronic, relapsing multi-organ neutrophilic/cytokine-driven inflammation plus progressive bone-marrow failure and clonal evolution to MDS/plasma-cell disease.

Molecular pathways / GO suggestions: - GO:0016567 protein ubiquitination (DECREASED) — the core lesion - GO:0000209 protein polyubiquitination - GO:0030968 endoplasmic reticulum unfolded protein response (INCREASED) - GO:0006914 autophagy (dysregulated) - GO:0032606 type I interferon production / GO:0034340 response to type I interferon (INCREASED) - GO:0070423 nucleotide-binding oligomerization domain containing signaling / GO:0140447 cytokine precursor processing (inflammasome) (INCREASED) - GO:0043123 positive regulation of canonical NF-κB signaling (INCREASED) - GO:0097190 apoptotic signaling / RIPK1-dependent necroptosis (INCREASED)

Cell types (CL suggestions): - CL:0000576 monocyte (key dysregulated effector) - CL:0000775 neutrophil (neutrophilic dermatosis, alveolitis) - CL:0000037 hematopoietic stem cell (clonal origin) - CL:0000839 myeloid lineage restricted progenitor cell - CL:0000764 erythroid lineage cell (vacuolated precursors) / CL:0000557 granulocyte monocyte progenitor cell - CL:0000786 plasma cell (associated dyscrasia)

Subcellular (GO cellular component): GO:0005783 endoplasmic reticulum; GO:0005829 cytosol (site of lost UBA1b activity); GO:0000502 proteasome complex.

Immune involvement: Prototypic autoinflammatory (innate-driven) disease, not classic autoimmunity — though autoantibody/overlap features occur. Cytokine drivers: IL-6, IL-1β, TNF-α, type I/II IFN.

Molecular profiling: Transcriptomics of patient marrow/blood shows interferon + inflammatory signatures arising early in primitive HSPCs and the myeloid lineage (Cell Reports Med / iScience 2023; PMC12092610, S2666379123003130). Single-cell genotype–phenotype mapping links the mutant clone directly to the inflammatory program and suggests therapeutic vulnerabilities (biorxiv 2024.05.19.594376). (IN_VITRO / COMPUTATIONAL)


7. Anatomical Structures Affected

Primary site: Bone marrow / hematopoietic system — the origin and engine. UBERON: UBERON:0002371 (bone marrow), UBERON:0000178 (blood).

Multi-organ secondary involvement (UBERON): - Skin — UBERON:0002097 (skin of body) / UBERON:0000014 (zone of skin) - Cartilage — auricular UBERON:0001691 (external ear) / nasal cartilage UBERON:0001737 (laryngeal cartilage—approx.); cartilage tissue UBERON:0002418 - Eye — UBERON:0000970 (eye); sclera UBERON:0001773; orbit UBERON:0001697 - Lung — UBERON:0002048 (lung); pleura UBERON:0000175 - Blood vessels (veins) — UBERON:0001638 (vein); vasculature UBERON:0002049 - Joints — UBERON:0000465 (material anatomical entity—joint) / UBERON:0001485 (synovial joint approx.)

Body systems: hematopoietic/immune, integumentary, respiratory, cardiovascular (venous), musculoskeletal, ocular/visual, occasionally nervous (aseptic meningitis) and reproductive (orchitis).

Tissue/cell level: myeloid and erythroid bone-marrow precursors (vacuolated); circulating monocytes and neutrophils; dermal neutrophilic/histiocytoid infiltrates; cartilage perichondrial inflammation.

Subcellular: ER (UPR), cytosol (ubiquitylation failure), proteasome; characteristic cytoplasmic vacuoles.

Localization/laterality: Generally systemic and bilateral (e.g., bilateral auricular chondritis, periorbital edema), though skin and pulmonary lesions can be patchy/asymmetric.


8. Temporal Development

  • Onset: Adult/late-onset. Median ~66 y (IQR ~63–73); essentially never pediatric (somatic clonal acquisition with age). HPO onset: HP:0003581 (Adult onset) → HP:0003596 (Middle age onset)/late onset. Pattern usually insidious/subacute with episodic flares.
  • Progression / stages: No formal staging. Conceptually: (1) early relapsing inflammatory phase often misdiagnosed as a rheumatologic syndrome → (2) glucocorticoid-dependent chronic inflammation with emerging cytopenias → (3) progressive marrow failure / transfusion dependence and clonal evolution (MDS, plasma-cell disease) → (4) end-stage cytopenias, infection, or transformation.
  • Course: Chronic, relapsing-remitting with cumulative organ damage; lifelong. Spontaneous durable remission is rare; remissions are typically treatment-induced (steroids, JAK inhibitors, hypomethylating agents) or curative only via allogeneic transplant.
  • Critical window: Earlier molecular diagnosis (recognizing VEXAS behind "relapsing polychondritis / Sweet / MDS in an older man") opens the window for clone-directed therapy and transplant evaluation before irreversible marrow failure.

9. Inheritance and Population

Epidemiology. - Prevalence (landmark genome-first study, Geisinger MyCode, 163,096 unselected adults): ~1 in 4,269 men >50 y and ~1 in 26,238 women >50 y; ~1 in 13,591 unrelated individuals >50 y overall.

"...estimated prevalence of disease-associated UBA1 variants... 1 in 4269 men and 1 in 26,238 women older than 50 years." — Beck DB et al., JAMA 2023;329(4):318-324 (PMID:36692560). (HUMAN_CLINICAL)

  • This reframed VEXAS from "ultra-rare" to a relatively common cause of unexplained adult inflammation in older men, almost certainly under-diagnosed. Incidence figures are not yet firmly established — (data gap).

Genetics of transmission. - Inheritance pattern: Not inherited — somatic/acquired. Functionally X-linked in the sense that the male single-X dosage explains the strong sex skew, but there is no germline transmission to offspring and no recurrence risk in families. - Penetrance: Among carriers identified genome-first, penetrance of the combined inflammatory+hematologic phenotype was reported as high (approaching ~100% in symptomatic ascertainment), though milder/oligosymptomatic carriers are increasingly recognized. - Expressivity: Highly variable (chondritis-predominant vs skin-predominant vs MDS-predominant), partly by genotype. - Anticipation / germline mosaicism / founder effects / consanguinity / carrier frequency: Not applicable (somatic disease).

Demographics. - Sex ratio: Strongly male; ~96% male / ~4% female (females usually require monosomy X or skewed XCI). - Age distribution: Overwhelmingly >50 y; peak 6th–8th decades. - Ethnic/geographic distribution: Reported worldwide across ancestries; no strong ethnic predilection established (the major cohorts are US and European). No endemic geography (not environmental/infectious).


10. Diagnostics

Definitive test — molecular. - UBA1 somatic mutation detection in peripheral blood and/or bone marrow (myeloid-enriched fractions increase sensitivity). Methods: targeted Sanger (high-VAF), NGS panels, ddPCR, or WGS/WES (caution: high-VAF somatic UBA1 can be misread as hemizygous germline on exome — PMID:36038944). Confirm somatic status by absence in skin fibroblasts/non-hematopoietic tissue.

Morphologic clue. - Bone marrow aspirate: cytoplasmic vacuoles in myeloid and erythroid precursor cells — the original "V." Highly suggestive but not 100% specific/sensitive.

Laboratory. - Persistently elevated CRP/ESR; macrocytic anemia (high MCV), variable thrombocytopenia/leukopenia/monocytopenia; ferritin often high. LOINC: CRP (LOINC:1988-5), ESR (LOINC:4537-7), MCV (LOINC:787-2), Hemoglobin (LOINC:718-7). - SPEP/immunofixation for monoclonal protein (plasma-cell dyscrasia screen).

Imaging. CT chest for pulmonary infiltrates/effusions; vascular imaging for VTE; cross-sectional imaging for large-vessel vasculitis when GCA/large-vessel overlap suspected.

Histopathology. Skin/marrow biopsy: neutrophilic/leukocytoclastic infiltrates, perichondrial inflammation; marrow shows myeloid hyperplasia ± dysplasia and vacuolated precursors.

Diagnostic criteria. No validated formal criteria yet. Working approach (GeneReviews; Koster/Mayo and others): adult male with relapsing multisystem inflammation (chondritis/skin/eye/lung) + macrocytic anemia/cytopenias ± marrow vacuoles + steroid dependence → test UBA1. Proposed clinical screening scores exist (e.g., to prioritize who to sequence) but are not consensus-finalized — (data gap / evolving).

Differential diagnosis (to distinguish): relapsing polychondritis, Sweet syndrome, polyarteritis nodosa, giant cell arteritis/large-vessel vasculitis, adult-onset Still disease, MDS without autoinflammation, IgG4-related disease, Behçet disease. The unifying discriminator is the somatic UBA1 mutation + marrow vacuoles + macrocytic anemia in an older man.

Screening. No population newborn/carrier screening (somatic disease). Emerging concept: opportunistic UBA1 testing in older men presenting with otherwise-unexplained relapsing inflammation plus macrocytosis.


11. Outcome / Prognosis

  • Mortality / survival: High. Estimated 5-year mortality up to ~50% from symptom onset in early cohorts; the discovery cohort reported 10/25 deaths.

"Of the 25 patients, 10 died during the study period." — Beck DB et al., NEJM 2020 (PMID:33108101). (HUMAN_CLINICAL)

  • Genotype-stratified 5-yr survival: p.Met41Leu ~100% > p.Met41Thr ~83% > p.Met41Val ~60–77% (Ferrada/Beck, Blood 2022, PMID:35793465).
  • Disease-specific mortality drivers: progressive cytopenias/marrow failure, infection (compounded by immunosuppression), thromboembolism, transformation to MDS/AML or progressive plasma-cell disease.
  • Prognostic factors: p.Met41Val genotype and transfusion dependence predict worse survival; ear chondritis associates with better prognosis; co-mutations in myeloid-malignancy genes worsen outcome; age and comorbidity matter.
  • Morbidity: Substantial — chronic steroid toxicity (osteoporosis, diabetes, infection), transfusion dependence, recurrent thrombosis, cumulative organ damage. Most patients fail to achieve durable drug-free remission.
  • Recovery potential: No spontaneous cure; allogeneic HSCT is the only potentially curative option and can eradicate the mutant clone, at the cost of significant transplant-related morbidity/mortality.

12. Treatment

No regulatory-approved therapy and no consensus guideline exist; management is empirical, drawn from cohorts/case series. Two strategic arms: (A) suppress inflammation and (B) target/eradicate the UBA1-mutant clone.

A. Anti-inflammatory / immunosuppressive - Glucocorticoids — first-line, almost universally effective but disease is steroid-dependent; chronic toxicity drives the need for steroid-sparing agents. MAXO: MAXO:0000058 (pharmacotherapy) / corticosteroid; CHEBI:50858 (corticosteroid) / CHEBI:8378 (prednisone). - JAK inhibitorsruxolitinib is the most effective JAK inhibitor (superior to tofacitinib/baricitinib/upadacitinib), with meaningful clinical response in roughly half of treated patients.

"Ruxolitinib is more effective than other JAK inhibitors to treat VEXAS syndrome." — Heiblig M et al., Blood 2022 (PMID:35609174). (HUMAN_CLINICAL) CHEBI:75045 (ruxolitinib); modality SMALL_MOLECULE; target JAK1/JAK2. - IL-6 inhibition (tocilizumab) — partial benefit (~26% response). CHEBI/NCIT tocilizumab; modality MONOCLONAL_ANTIBODY. - IL-1 inhibition (anakinra, canakinumab) — limited efficacy (<10%); anakinra can cause severe injection-site reactions in VEXAS. - Conventional DMARDs (methotrexate, azathioprine), TNF inhibitors — generally poorly/inconsistently effective.

B. Clone-directed (hematologic) - Hypomethylating agents — azacitidine — clinical responses (~5/11 with concurrent MDS in GeneReviews summary) and, importantly, occasional deep/complete molecular remission of the UBA1 clone, sometimes permitting therapy de-escalation.

"Two patients achieved complete molecular remission of the underlying UBA1 mutant clone... receiving treatment with the hypomethylating agent azacitidine." — Blood / Annals of Hematology 2023–2025 reports. (HUMAN_CLINICAL) CHEBI:2038 (azacitidine); MAXO chemotherapy/pharmacotherapy. - Allogeneic hematopoietic stem cell transplantation (allo-HSCT) — the only curative therapy; eradicates the mutant clone. Systematic review/meta-analysis supports efficacy in selected, fit patients, balanced against transplant-related mortality (Nature BMT 2024, s41409-024-02375-3). MAXO: MAXO:0001175/MAXO:0010039 (hematopoietic/organ transplantation); modality CELL_THERAPY.

Emerging / experimental. UBA1-targeted and clone-selective strategies, optimized HMA + JAKi combinations, and refined transplant conditioning are under active study. Recent retrospective treatment-outcome cohorts (Lancet Rheumatology 2025, PIIS2665-9913(25)00034-7) are defining comparative effectiveness. Relevant trial registries: search ClinicalTrials.gov for "VEXAS" (e.g., natural-history/genetics protocol NCT06004349; several interventional JAKi/HMA studies). (Add specific NCT IDs at curation time.)

Supportive care. Transfusion support, infection prophylaxis (especially under steroids/JAKi/HMA — PJP prophylaxis), anticoagulation for VTE, bone protection, vaccination. MAXO:0000950 (supportive care).

Pharmacogenomics. No VEXAS-specific PGx; standard JAKi/azacitidine considerations apply.


13. Prevention

  • Primary prevention: None possible — disease arises from a random somatic mutation in aging hematopoiesis; no modifiable exposure, no vaccine.
  • Secondary prevention (early detection): The highest-yield "prevention" is earlier diagnosis — testing UBA1 in older men with unexplained relapsing inflammation + macrocytic anemia to intervene before marrow failure. Genome-first ascertainment (PMID:36692560) shows latent/under-recognized cases exist.
  • Tertiary prevention (complications): VTE prophylaxis/anticoagulation, infection prophylaxis during immunosuppression, steroid-toxicity mitigation (bone, glucose), transfusion-iron management, and timely transplant referral to prevent clonal progression.
  • Genetic counseling: Reassurance that VEXAS is somatic and not heritable — no offspring/sibling recurrence risk, no prenatal/carrier testing indicated. This is an important counseling point distinguishing it from germline autoinflammatory syndromes.
  • Public-health/environmental interventions: Not applicable.

14. Other Species / Natural Disease

  • Taxonomy: Human disease (NCBITaxon:9606). No naturally occurring animal counterpart described.
  • Orthologous gene: Uba1 is highly conserved — mouse Uba1 (NCBI Gene 22201), zebrafish uba1. Strong evolutionary conservation of the ubiquitin-activation step makes the mechanism studyable across species.
  • Natural disease in animals (OMIA/veterinary): None reported — (data gap / not applicable). There is no spontaneous companion-animal or wildlife VEXAS analog on record.
  • Comparative biology: The disease itself is human-specific (requires the human UBA1b cytoplasmic-isoform start-codon architecture at Met41 plus age-related clonal hematopoiesis); engineered animal models (below) are the route to cross-species mechanistic study.
  • Transmission/zoonosis: Not applicable (non-communicable, somatic).

15. Model Organisms

  • Zebrafish (Danio rerio): uba1-perturbation models recapitulate IRF3 accumulation, excessive type I interferon, and inflammation, supporting the proximal-ubiquitylation→IFN mechanism. (MODEL_ORGANISM) — useful for innate-immune readouts and drug screening. ZFIN resource.
  • Mouse (Mus musculus): Conditional/hematopoietic Uba1-mutant or knockdown models show UPR activation and myeloid bias, with recent work dissecting inflammation vs myeloid-bias as partly independent of RIPK3–CASP8 (Nature 2025, s41586-025-09815-0). (MODEL_ORGANISM) MGI resource; IMPC for Uba1 alleles.
  • In vitro / cellular: Patient-derived monocytes/macrophages and CD34+ HSPCs, iPSC-derived myeloid cells, and engineered Met41-mutant cell lines reproduce reduced ubiquitylation, ER/UPR stress, inflammasome activation, and RIPK1-mediated death. (IN_VITRO) — workhorse systems for mechanism and therapeutic-vulnerability screens (single-cell genotype–phenotype mapping, biorxiv 2024.05.19.594376).
  • Phenotype recapitulation: Models reproduce the molecular/inflammatory arms well (ubiquitylation defect, UPR, IFN/inflammasome, myeloid skewing).
  • Limitations: No single model fully reproduces the multi-organ relapsing clinical syndrome (chondritis, skin, vacuolated precursors, MDS evolution) seen in patients; the age-dependent somatic-clonal acquisition and the human-specific UBA1b isoform context are hard to mimic. Treat model→human translation as a HUMAN_MODEL_MISMATCH candidate where mouse/zebrafish data inform mechanism but human-disease fidelity remains open.
  • Resources: MGI, IMPC, ZFIN, Cellosaurus (patient/iPSC lines), GEO (patient transcriptomics).

Key Citations (PMID-anchored)

Claim Reference PMID Evidence type
Discovery; UBA1 p.Met41 somatic mutation; vacuoles; 25 men; 10 deaths Beck DB et al. NEJM 2020;383:2628-2638 33108101 HUMAN_CLINICAL + IN_VITRO
Population prevalence (1/4269 men >50) Beck DB et al. JAMA 2023;329:318-324 36692560 HUMAN_CLINICAL
Cytoplasmic UBA1b translation; genotype–survival (Val worst) Ferrada/Beck et al. Blood 2022;140:1496-1506 35793465 IN_VITRO + HUMAN_CLINICAL
Novel/expanded UBA1 variant spectrum (splice, non-Met41) Poulter JA et al. Blood 2021;137:3676-3681 33690795 HUMAN_CLINICAL
Ruxolitinib superior among JAK inhibitors Heiblig M et al. Blood 2022 35609174 HUMAN_CLINICAL
Exome can misread high-VAF somatic UBA1 as hemizygous (case report) 36038944 HUMAN_CLINICAL
Comprehensive clinical/genetic synthesis GeneReviews: VEXAS Syndrome (Beck DB) Bookshelf NBK614471 Review
Mechanism: inflammation vs myeloid bias independent Nature 2025 (s41586-025-09815-0) (PMID pending) MODEL_ORGANISM

Sources (web): - Beck et al. NEJM 2020 — PMID:33108101 - Beck et al. JAMA 2023 — PMID:36692560 - GeneReviews: VEXAS Syndrome — NBK614471 - OMIM #301054 - Ferrada/Beck Blood 2022 — Translation of cytoplasmic UBA1 (PMC9523373) - Heiblig et al. Blood 2022 — Ruxolitinib (PMID:35609174) - Nature 2025 — Independent mechanisms of inflammation and myeloid bias - NCI/DCEG genome-first prevalence summary - Bone Marrow Transplantation 2024 — allo-HSCT meta-analysis - Lancet Rheumatology 2025 — treatment outcomes cohort


Curation notes for the dismech entry (kb/disorders/VEXAS_Syndrome.yaml)

  • Category: Complex — clean fit; this is a clonal-hematopoietic autoinflammatory disorder bridging rheumatology and hematology.
  • MONDO: MONDO:0026777 · Gene: hgnc:12469 (UBA1) · note somatic origin in the genetic block (GENO somatic mutation, not germline inheritance).
  • Pathophysiology causal chain to encode: UBA1b loss → ↓cytoplasmic ubiquitylation (GO:0016567 DECREASED) → ER/UPR stress (GO:0030968 INCREASED) → inflammasome/NF-κB/type-I-IFN (GO:0034340, GO:0043123 INCREASED) → myeloid-biased dysplastic hematopoiesis + multi-organ neutrophilic inflammation.
  • Module conformance candidates: This is a natural fit for an autoinflammation / innate-immune-dysregulation pattern; if a "clonal hematopoiesis" or "type-I-interferonopathy"-adjacent module exists or is created, link it. (No exact existing module from the CLAUDE.md list maps cleanly — flag as a possible new-module opportunity rather than forcing a fit.)
  • Before committing evidence: every PMID above must be just fetch-reference'd and every snippet: verified as an exact substring of the real abstract (the quotes here are paraphrase-adjacent search excerpts and must be replaced with verified verbatim text). Run just validate, just validate-references, and just validate-terms-file on the file.
  • Data gaps flagged: ICD-11 code; precise incidence; QoL instrument data; epigenome studies; animal natural-disease (OMIA); finalized formal diagnostic criteria. Consider discussions with kind: KNOWLEDGE_GAP for these, and kind: HUMAN_MODEL_MISMATCH for the model-organism translational gap.